SCHEMBL23854259

SCHEMBL23854259

O=C(O)/C=C/c1ccc(CCc2ccccc2)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.67
HDAC1 Q13547 3/20 0.67
HDAC2 Q92769 3/20 0.67
HDAC8 Q9BY41 3/20 0.67
HCAR2 Q8TDS4 2/20 0.67
HDAC4 P56524 2/20 0.67
HDAC7 Q8WUI4 2/20 0.67
HDAC10 Q969S8 2/20 0.67
HDAC11 Q96DB2 2/20 0.67
HDAC6 Q9UBN7 2/20 0.67
HDAC9 Q9UKV0 2/20 0.67
HDAC5 Q9UQL6 2/20 0.67
TNKS O95271 1/20 0.67
TNKS2 Q9H2K2 1/20 0.67
TBXAS1 P24557 2/20 0.58
FFAR1 O14842 2/20 0.58
AKR1B10 O60218 4/20 0.57
AKR1B1 P15121 4/20 0.57
ESR1 P03372 2/20 0.57
ESR2 Q92731 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3225302 1.00 HDAC3 (0.67) HDAC3HDAC1HDAC2HDAC8HCAR2
Cinnamic Acid SCHEMBL890441 0.94 HCAR2 (0.76) HDAC3HDAC1HDAC2HDAC8HCAR2
SCHEMBL3105287 0.93 HDAC1 (0.62) HDAC3HDAC1HDAC2HDAC8HCAR2
SCHEMBL3688787 0.93 HDAC1 (0.62) HDAC3HDAC1HDAC2HDAC8HCAR2
SCHEMBL3105298 0.93 HDAC1 (0.62) HDAC3HDAC1HDAC2HDAC8HCAR2
SCHEMBL2772402 0.89 TBXAS1 (0.71) HDAC3HDAC1HDAC2HDAC8HCAR2
SCHEMBL459101 0.89 TBXAS1 (0.71) HDAC3HDAC1HDAC2HDAC8HCAR2
Cinnamic Acid SCHEMBL28536919 0.86 HCAR2 (0.63) HDAC3HDAC1HDAC2HDAC8HCAR2
SCHEMBL11827873 0.85 RAB9A (0.56) HDAC3HDAC1HDAC2HDAC8HCAR2
SCHEMBL28087116 0.85 AKR1B10 (0.53) HDAC3HDAC1HDAC2HDAC8HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11307508-B2 Electrophotographic photoreceptor, process cartridge, and image forming apparatus FUJIFILM BUSINESS INNOVATION CORP. (JP) 2022-04-19 US disclosed
US-20210302848-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, PROCESS CARTRIDGE, AND IMAGE FORMING APPARATUS FUJI XEROX CO., LTD. (JP) 2021-09-30 US disclosed