SCHEMBL2386287

SCHEMBL2386287

COC(=O)[C@H](Cc1ccccc1)N(N[C@@H](Cc1cccc(O)c1)C(=O)O)C(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 2/20 0.45
ITGB7 P26010 2/20 0.45
ACE P12821 1/20 0.43
KLK5 Q9Y337 1/20 0.43
NOS2 P35228 1/20 0.42
NLRP3 Q96P20 1/20 0.40
APP P05067 1/20 0.39
MDM4 O15151 1/20 0.39
MDM2 Q00987 1/20 0.39
PTPN1 P18031 1/20 0.39
CTSS P25774 3/20 0.39
CTSB P07858 2/20 0.39
CTSK P43235 2/20 0.39
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.38
CTSL P07711 1/20 0.38
MAOA P21397 1/20 0.38
YAP1 P46937 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2387887 0.92 ITGA4 (0.42) ITGA4ITGB7ACEKLK5NOS2
SCHEMBL2385485 0.92 ITGA4 (0.49) ITGA4ITGB7ACEKLK5APP
SCHEMBL2385950 0.91 ITGA4 (0.47) ITGA4ITGB7ACEKLK5MDM4
SCHEMBL2386456 0.90 POLB (0.44) ITGA4ITGB7ACEKLK5PTPN1
SCHEMBL2386802 0.89 POLB (0.46) ITGA4ITGB7ACEKLK5MEN1
SCHEMBL2388163 0.89 NOS2 (0.44) NOS2NLRP3MDM4MDM2ALDH1A1
SCHEMBL2386579 0.89 GPR132 (0.48) ITGA4ITGB7ACEPTPN1YAP1
SCHEMBL2386292 0.89 ITGA4 (0.42) ITGA4ITGB7ACEKLK5CTSS
SCHEMBL2384997 0.88 USP2 (0.43) ITGA4ITGB7ACEKLK5NOS2
SCHEMBL2384999 0.87 POLB (0.43) ITGA4ITGB7ACEKLK5PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8017378-B2 Method for production of optically active biphenylalanine compound or salt or ester thereof SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2011-09-13 US disclosed
US-20090011475-A1 Method For Production of Optically Active Biphenylalanine Compound or Salt or Ester Thereof SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2009-01-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090011475-A1 Method For Production of Optically Active Biphenylalanine Compound or Salt or Ester Thereof DNPEP, APEH, PAH ITGA4 4819/4885ITGB7 4625/4885ACE 31/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.