SCHEMBL23872467

SCHEMBL23872467

CNc1ccnc2c1ccn2CC(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.34
CYP1A2 P05177 1/20 0.34
HTR3A P46098 5/20 0.33
GRM1 Q13255 4/20 0.33
METAP2 P50579 1/20 0.33
SLC40A1 Q9NP59 1/20 0.32
BMPR1B O00238 1/20 0.32
ACVR1B P36896 1/20 0.32
TGFBR1 P36897 1/20 0.32
ACVRL1 P37023 1/20 0.32
ACVR1 Q04771 1/20 0.32
PIK3CA P42336 1/20 0.31
MTOR P42345 1/20 0.31
FGFR1 P11362 1/20 0.31
FGFR4 P22455 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29324232 0.78 CYP17A1 (0.35) CYP17A1CYP1A2HTR3APIK3CAMTOR
SCHEMBL30098893 0.76 HTR6 (0.42) HTR3AMETAP2
SCHEMBL23858812 0.74 HTR3A (0.44) HTR3AMETAP2SLC40A1PIK3CAMTOR
SCHEMBL23771391 0.73 UTS2R (0.38) GRM1SLC40A1
SCHEMBL23872096 0.72 HTR3A (0.40) HTR3AMETAP2PIK3CAMTOR
SCHEMBL24229270 0.71 SLC40A1 (0.36) GRM1SLC40A1
SCHEMBL24376134 0.71 SLC40A1 (0.36) GRM1SLC40A1
Potassium Ion SCHEMBL23858590 0.70 HTR3A (0.39) CYP17A1CYP1A2HTR3APIK3CAMTOR
SCHEMBL22133201 0.70 SLC40A1 (0.38) GRM1SLC40A1
SCHEMBL20971252 0.66 HPRT1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021191359-A1 MONOACYLGLYCEROL LIPASE MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2021-09-30 WO disclosed