SCHEMBL23891742

SCHEMBL23891742

CC(=O)CN1C(=O)OC2(CC3(CC3)c3cc(C)ccc32)C1=O

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
EP300 Q09472 10/20 0.34
CREBBP Q92793 4/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2C8 P10632 1/20 0.33
CYP2C9 P11712 1/20 0.33
BDKRB2 P30411 1/20 0.33
POLB P06746 1/20 0.33
GABRA1 P14867 1/20 0.33
SLC6A4 P31645 1/20 0.33
HTR2B P41595 1/20 0.33
SLC6A3 Q01959 1/20 0.33
TMEM97 Q5BJF2 1/20 0.33
PLK3 Q9H4B4 1/20 0.33
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23891729 0.89 EP300 (0.33) EP300CREBBPCYP3A4CYP2C8CYP2C9
SCHEMBL23891672 0.85 CCKBR (0.34) NPC1RAB9AEP300CREBBPCYP3A4
SCHEMBL23891707 0.83 EP300 (0.49) EP300CREBBPCYP3A4CYP2C8CYP2C9
SCHEMBL23891583 0.71 EP300 (0.46) EP300CREBBPCYP3A4CYP2C8CYP2C9
SCHEMBL24350741 0.70 EP300 (0.46) EP300CREBBPCYP3A4CYP2C8CYP2C9
SCHEMBL23891727 0.70 EP300 (0.45) EP300CREBBPCYP3A4CYP2C8CYP2C9
SCHEMBL23891706 0.70
SCHEMBL23891650 0.70 CYP3A4 (0.35) CYP3A4POLB
SCHEMBL23891578 0.70 CYP3A4 (0.35) CYP3A4POLB
SCHEMBL23891728 0.68 CYP3A4 (0.34) CREBBPCYP3A4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3889138-A1 HISTONE ACETYLASE P300 INHIBITOR AND USE THEREOF Hinova Pharmaceuticals Inc. (CN) 2021-10-06 EP disclosed