SCHEMBL2390105

SCHEMBL2390105

C#Cc1ccc(C#N)c(F)c1

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 2/20 0.53
CYP11B2 P19099 17/20 0.45
CYP11B1 P15538 16/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24942536 0.85 CYP11B2 (0.55) TRPV4CYP11B2CYP11B1
SCHEMBL16182687 0.85 HDAC8 (0.34) TRPV4CYP11B2CYP11B1
SCHEMBL1797379 0.85 TRPV4 (0.59) TRPV4CYP11B2CYP11B1
SCHEMBL3633872 0.83 TRPV4 (0.41) TRPV4CYP11B2CYP11B1
SCHEMBL15577767 0.83 TRPV4 (0.44) TRPV4CYP11B2CYP11B1
SCHEMBL9612005 0.81 TRPV4 (0.55) TRPV4CYP11B2CYP11B1
SCHEMBL4394514 0.80 MAOB (0.39) TRPV4
SCHEMBL16961654 0.79 TRPV4 (0.53) TRPV4CYP11B2CYP11B1
SCHEMBL1914223 0.78 MAOA (0.34) TRPV4
SCHEMBL14183919 0.75 TSHR (0.45) CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11829021-B2 Polymer dispersed liquid crystal display device comprising a polymer network having a helical structure and method for manufacturing the same Sharp Display Technology Corporation (JP) 2023-11-28 US disclosed
US-20230205010-A1 LIQUID CRYSTAL DISPLAY ELEMENT Sharp Display Technology Corporation (JP) 2023-06-29 US disclosed
US-20230024383-A1 LIQUID CRYSTAL DISPLAY DEVICE Sharp Display Technology Corporation (JP) 2023-01-26 US disclosed
WO-2016055947-A1 ALKYNE COMPOUNDS AS S-NITROSOGLUTATHIONE REDUCTASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2016-04-14 WO disclosed
US-8013001-B2 Modulators of LXR EXELIXIS, INC. (US) 2011-09-06 US disclosed
US-8013001-B2 Modulators of LXR EXELIXIS, INC. (US) 2011-09-06 US disclosed
US-20100056582-A1 Modulators of LXR X-CEPTOR THERAPEUTICS, INC. (US) 2010-03-04 US disclosed
US-20100056582-A1 Modulators of LXR X-CEPTOR THERAPEUTICS, INC. (US) 2010-03-04 US disclosed
US-7482366-B2 Modulators of LXR X-CEPTOR THERAPEUTICS, INC. (US) 2009-01-27 US disclosed
US-7482366-B2 Modulators of LXR X-CEPTOR THERAPEUTICS, INC. (US) 2009-01-27 US disclosed
US-20080119488-A1 Modulators Of Nuclear Receptors EXELIXIS, INC. (US) 2008-05-22 US disclosed
US-20080119488-A1 Modulators Of Nuclear Receptors EXELIXIS, INC. (US) 2008-05-22 US disclosed
EP-1773337-A2 MODULATORS OF NUCLEAR RECEPTORS Exelixis, Inc. (US) 2007-04-18 EP disclosed
WO-2006025979-A9 MODULATORS OF NUCLEAR RECEPTORS EXELIXIS INC (US) 2006-04-20 WO disclosed
WO-2006025979-A2 MODULATORS OF NUCLEAR RECEPTORS EXELIXIS, INC. (US) 2006-03-09 WO disclosed
US-20050080111-A1 Modulators of LXR X-CEPTOR THERAPEUTICS, INC. (US) 2005-04-14 US disclosed
EP-0648723-B1 Diphenylacetylene compound, process for preparing the same and liquid crystal composition and element comprising the same SUMITOMO CHEMICAL CO (JP) 1998-05-20 EP disclosed
US-5725797-A Silacyclohexane compound, a process for producing the same, and a liquid crystal composition comprising the same SHIN-ETSU CHEMICAL CO., LTD. (JP) 1998-03-10 US disclosed
US-5658489-A EXCELLENT ANISOTROPY OF REFRACTIVE INDEX; LOW VISCOSITY SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-08-19 US disclosed
EP-0648723-A1 Diphenylacetylene compound, process for preparing the same and liquid crystal composition and element comprising the same SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1995-04-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080119488-A1 Modulators Of Nuclear Receptors NR1H2, NR0B1, NR1H3 TRPV4 2034/4885CYP11B2 58/4885CYP11B1 42/4885
US-20050080111-A1 Modulators of LXR NR1H2, NR1H3, NR1H4 TRPV4 3079/4885CYP11B2 85/4885CYP11B1 34/4885
US-20100056582-A1 Modulators of LXR NR1H2, NR1H3, NR1H4 TRPV4 3079/4885CYP11B2 85/4885CYP11B1 34/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.