SCHEMBL23904802

SCHEMBL23904802

CC1(CO)COc2c1cc(C(=O)C(F)(F)F)nc2-c1ccc(F)cc1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CFTR P13569 4/20 0.36
DHODH Q02127 1/20 0.34
IDO1 P14902 3/20 0.33
CYP2C9 P11712 2/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
MAP2K4 P45985 1/20 0.33
PTGDR2 Q9Y5Y4 2/20 0.32
KCNH2 Q12809 2/20 0.32
DPP4 P27487 2/20 0.31
GRM2 Q14416 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
SCN9A Q15858 1/20 0.31
CYP3A4 P08684 1/20 0.31
NTRK1 P04629 1/20 0.31
NTRK2 Q16620 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23905462 0.92 CFTR (0.36) CFTRDHODHIDO1CYP2C9HDAC4
SCHEMBL23905699 0.88 CFTR (0.32) CFTRIDO1CYP2C9
SCHEMBL23905327 0.87 CFTR (0.34) CFTRMAP2K4PTGDR2KCNH2
SCHEMBL23904788 0.86 DPP4 (0.32) CFTRIDO1CYP2C9PTGDR2DPP4
SCHEMBL23905340 0.86 CFTR (0.33) CFTRDHODHHDAC4HDAC1HDAC6
SCHEMBL23905333 0.84 MAP2K4 (0.32) CFTRDHODHHDAC4HDAC1HDAC6
SCHEMBL23905338 0.84 MAP2K4 (0.32) CFTRDHODHHDAC4HDAC1HDAC6
SCHEMBL23196085 0.83 GAA (0.35) CFTRDHODHPTGDR2
SCHEMBL23905342 0.83 MAP2K4 (0.34) CFTRDHODHHDAC4HDAC1HDAC6
SCHEMBL23905349 0.82 CFTR (0.33) CFTRDHODHHDAC4HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021198981-A1 ANTIVIRAL COMPOUNDS AND USES THEREOF Janssen Biopharma, Inc. (US) 2021-10-07 WO disclosed