SCHEMBL23905462

SCHEMBL23905462

CC1(CF)COc2c1cc(C(=O)C(F)(F)F)nc2-c1ccc(F)cc1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CFTR P13569 4/20 0.36
MAP2K4 P45985 1/20 0.33
KCNH2 Q12809 2/20 0.32
DHODH Q02127 1/20 0.32
CYP2C9 P11712 1/20 0.32
IDO1 P14902 1/20 0.32
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
GRM2 Q14416 1/20 0.31
CYP3A4 P08684 1/20 0.31
NTRK1 P04629 1/20 0.31
NTRK2 Q16620 1/20 0.31
TRPV1 Q8NER1 2/20 0.30
PTGDR2 Q9Y5Y4 2/20 0.30
CTSA P10619 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA2B P29275 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23904802 0.92 CFTR (0.36) CFTRMAP2K4KCNH2DHODHCYP2C9
SCHEMBL23905463 0.88 CFTR (0.32) CFTR
SCHEMBL23905342 0.87 MAP2K4 (0.34) CFTRMAP2K4DHODHHDAC4HDAC1
SCHEMBL23905327 0.87 CFTR (0.34) CFTRMAP2K4KCNH2PTGDR2CTSA
SCHEMBL23905349 0.86 CFTR (0.33) CFTRMAP2K4DHODHHDAC4HDAC1
SCHEMBL23905333 0.84 MAP2K4 (0.32) CFTRMAP2K4KCNH2DHODHHDAC4
SCHEMBL23905339 0.84 MAP2K4 (0.32) CFTRMAP2K4HDAC4HDAC1HDAC6
SCHEMBL23196085 0.83 GAA (0.35) CFTRDHODHPTGDR2CTSAADORA2A
SCHEMBL23196082 0.83 HDAC4 (0.38) CFTRCYP2C9HDAC4HDAC6CYP3A4
SCHEMBL23905340 0.82 CFTR (0.33) CFTRMAP2K4KCNH2DHODHHDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021198981-A1 ANTIVIRAL COMPOUNDS AND USES THEREOF Janssen Biopharma, Inc. (US) 2021-10-07 WO disclosed