SCHEMBL23905616

SCHEMBL23905616

C[C@]1(C(=O)NC2CC2)COc2c1cc(C(O)(CN)C(F)(F)F)nc2-c1ccc(F)cc1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.36
GABRA5 P31644 5/20 0.33
RORC P51449 3/20 0.32
CYP2C8 P10632 2/20 0.32
CYP2C9 P11712 2/20 0.32
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
CFTR P13569 3/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
GRIN2B Q13224 2/20 0.31
RXFP1 Q9HBX9 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23905374 0.90 CFTR (0.33) GABRA5CYP2C9CFTRCYP3A4
SCHEMBL23905533 0.90 CFTR (0.33) GABRA5CYP2C9CFTRCYP3A4
SCHEMBL23905693 0.88 GABRA5 (0.33) DPP4GABRA5RORCCYP2C8CYP2C9
SCHEMBL23904871 0.87 CFTR (0.33) CFTRPTGS2CYP3A4
SCHEMBL31412435 0.87 CFTR (0.33) CFTRPTGS2CYP3A4
SCHEMBL23905407 0.87 CFTR (0.33) CFTRPTGS2CYP3A4
SCHEMBL23905581 0.87 CFTR (0.33) CFTRPTGS2CYP3A4
SCHEMBL24986093 0.87 CFTR (0.41) RORCCYP2C9CFTRCYP3A4
SCHEMBL23904755 0.86 CFTR (0.33) CYP2C9CFTR
SCHEMBL23904764 0.86 CFTR (0.33) CYP2C9CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021198981-A1 ANTIVIRAL COMPOUNDS AND USES THEREOF Janssen Biopharma, Inc. (US) 2021-10-07 WO disclosed