SCHEMBL23906394

SCHEMBL23906394

O=C(O)CN1CCC2(CC(OI)C2)C1

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 4/20 0.37
ITGA2B P08514 4/20 0.37
FFAR1 O14842 1/20 0.34
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23896280 0.84 ITGB3 (0.37) ITGB3ITGA2BFFAR1HSD17B10
SCHEMBL23906396 0.81 ELANE (0.33) HSD17B10
SCHEMBL25547732 0.81 ITGB3 (0.35) ITGB3ITGA2BFFAR1HSD17B10
SCHEMBL25477017 0.81 ITGB3 (0.35) ITGB3ITGA2BFFAR1HSD17B10
SCHEMBL23906369 0.80 ITGB3 (0.40) ITGB3ITGA2BHSD17B10
SCHEMBL23968807 0.79 ITGB3 (0.40) ITGB3ITGA2BHSD17B10
SCHEMBL14671193 0.77 ITGB3 (0.42) ITGB3ITGA2BHSD17B10
SCHEMBL23968808 0.75 ITGB3 (0.37) ITGB3ITGA2BHSD17B10
SCHEMBL14671149 0.74 ITGB3 (0.43) ITGB3ITGA2BHSD17B10
SCHEMBL20793574 0.71 TSHR (0.42) ITGB3ITGA2BHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021203025-A1 1 H-PYRAZOLO[4,3-G]ISOQUINOLINE AND 1 H-PYRAZOLO[4,3-G]QUINOLINE DERIVATIVES AS ALPHA-1 -ANTITRYPSIN MODULATORS FOR TREATING ALPHA-1 -ANTITRYPSIN DEFICIENCY (AATD) VERTEX PHARMACEUTICALS INCORPORATED (US) 2021-10-07 WO disclosed