SCHEMBL23912247

SCHEMBL23912247

CCc1nc2cccc(/C=C/CC3CCCCC3)c2c(=O)n1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.46
HDAC8 Q9BY41 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
DRD1 P21728 4/20 0.43
DRD5 P21918 4/20 0.43
PDE7A Q13946 1/20 0.41
PIK3CD O00329 3/20 0.41
PIK3R1 P27986 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.39
ALDH1A1 P00352 1/20 0.39
KCNH2 Q12809 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
GAA P10253 1/20 0.37
ALOX15 P16050 1/20 0.37
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
USP2 O75604 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17458293 0.82 HDAC1 (0.47) HDAC1HDAC8HDAC6PIK3CDPIK3R1
SCHEMBL17458291 0.82 HDAC1 (0.47) HDAC1HDAC8HDAC6PIK3CDPIK3R1
SCHEMBL23912298 0.79 HDAC1 (0.52) HDAC1HDAC8HDAC6PIK3CDPIK3R1
SCHEMBL20404285 0.79 HDAC1 (0.50) HDAC1HDAC8HDAC6PIK3CDPIK3R1
SCHEMBL23912240 0.77 PIK3CD (0.55) HDAC6DRD1DRD5PDE7APIK3CD
SCHEMBL17461948 0.76 PIK3CD (0.43) HDAC1HDAC8HDAC6PIK3CDPIK3R1
SCHEMBL20404396 0.76 PIK3CD (0.57) PIK3CDPIK3R1SMN1; SMN2ALDH1A1KCNH2
SCHEMBL19916811 0.75 HDAC1 (0.51) HDAC1HDAC8HDAC6PIK3CDPIK3R1
SCHEMBL16597182 0.71 SMN1; SMN2 (0.50) PIK3CDPIK3R1SMN1; SMN2ALDH1A1KCNH2
SCHEMBL16597185 0.71 PDE10A (0.52) PIK3CDPIK3R1SMN1; SMN2ALDH1A1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3160960-B1 PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS GILEAD SCIENCES INC (US) 2021-10-13 EP disclosed