SCHEMBL20404285

SCHEMBL20404285

CCc1nc2cccc(C=O)c2c(=O)n1-c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.50
HDAC8 Q9BY41 2/20 0.50
HDAC6 Q9UBN7 2/20 0.50
ALDH1A1 P00352 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
ESR1 P03372 1/20 0.45
ESR2 Q92731 1/20 0.45
PIK3CD O00329 2/20 0.44
PIK3R1 P27986 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
MAPT P10636 1/20 0.42
USP2 O75604 1/20 0.42
KCNH2 Q12809 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42
LMNA P02545 1/20 0.42
MAPK1 P28482 1/20 0.42
PSMD14 O00487 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23912298 0.88 HDAC1 (0.52) HDAC1HDAC8HDAC6ALDH1A1SMN1; SMN2
SCHEMBL20404396 0.84 PIK3CD (0.57) ALDH1A1SMN1; SMN2NPC1RAB9AESR1
SCHEMBL16597185 0.82 PDE10A (0.52) ALDH1A1SMN1; SMN2NPC1RAB9AESR1
SCHEMBL17235505 0.82 ESR1 (0.60) HDAC1HDAC8HDAC6ALDH1A1SMN1; SMN2
SCHEMBL16597182 0.82 SMN1; SMN2 (0.50) ALDH1A1SMN1; SMN2NPC1RAB9AESR1
SCHEMBL23912253 0.81 SMN1; SMN2 (0.45) HDAC1HDAC8HDAC6ALDH1A1SMN1; SMN2
SCHEMBL20404284 0.80 SMN1; SMN2 (0.48) HDAC1HDAC8HDAC6ALDH1A1SMN1; SMN2
SCHEMBL19916811 0.79 HDAC1 (0.51) HDAC1HDAC8HDAC6ALDH1A1SMN1; SMN2
SCHEMBL21185366 0.79 PIK3CD (0.48) ALDH1A1SMN1; SMN2NPC1RAB9AESR1
SCHEMBL20247392 0.79 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2NPC1RAB9AESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2935246-B1 ISOQUINOLINONE OR QUINAZOLINONE PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS GILEAD CALISTOGA LLC (US) 2018-07-25 EP disclosed