SCHEMBL23916844

SCHEMBL23916844

Cc1cc(Cl)c2[nH]ccc2c1C(C)C

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 5/20 0.36
AXL P30530 2/20 0.35
PRKCI P41743 2/20 0.35
AURKA O14965 2/20 0.33
TPX2 Q9ULW0 2/20 0.33
AHR P35869 1/20 0.32
CFB P00751 2/20 0.32
NR3C1 P04150 1/20 0.32
PGR P06401 1/20 0.32
CCR8 P51685 1/20 0.31
LMNA P02545 1/20 0.31
KMT2A Q03164 1/20 0.31
MAPT P10636 1/20 0.30
PRKCQ Q04759 1/20 0.30
PRKCD Q05655 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27051645 0.88 AXL (0.34) P2RX7AXLPRKCIAURKATPX2
SCHEMBL20939366 0.79 P2RX7 (0.42) P2RX7AXLPRKCIAURKATPX2
SCHEMBL22328043 0.74 AXL (0.34) P2RX7AXLPRKCIAURKATPX2
SCHEMBL19420465 0.74 ACHE (0.39) P2RX7AXLPRKCIAURKATPX2
SCHEMBL1146475 0.73 P2RX7 (0.40) P2RX7AXLPRKCIAURKATPX2
SCHEMBL31549623 0.73 CFB (0.40) P2RX7AXLPRKCIAURKATPX2
SCHEMBL18683281 0.72 P2RX7 (0.38) P2RX7AXLPRKCIAURKATPX2
SCHEMBL1465882 0.71 AHR (0.42) P2RX7AXLPRKCIAURKATPX2
SCHEMBL12278257 0.70 AHR (0.38) P2RX7AXLPRKCIAHRCCR8
SCHEMBL26077500 0.70 AURKA (0.38) P2RX7AXLPRKCIAURKATPX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240025918-A1 KRAS G12D Inhibitors JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2024-01-25 US disclosed
US-20240025918-A1 KRAS G12D Inhibitors JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2024-01-25 US disclosed
US-20210317127-A1 HETEROCYCLIC SPIRO COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF CANCER ARAXES PHARMA LLC (US) 2021-10-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210317127-A1 HETEROCYCLIC SPIRO COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF CANCER KRAS, NRAS, HRAS P2RX7 3928/4885AXL 1914/4885PRKCI 379/4885
US-20240025918-A1 KRAS G12D Inhibitors KRAS, NRAS, HRAS P2RX7 3221/4885AXL 1347/4885PRKCI 234/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.