SCHEMBL23918335

SCHEMBL23918335

O=CCSc1nc2c(cnn2-c2ccccc2)c(=O)[nH]1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.75
TSHR P16473 2/20 0.75
MAPT P10636 2/20 0.66
CREBBP Q92793 2/20 0.66
HSD17B10 Q99714 2/20 0.66
L3MBTL1 Q9Y468 3/20 0.64
TP53 P04637 2/20 0.64
KMT2A Q03164 4/20 0.63
HPGD P15428 3/20 0.63
MEN1 O00255 3/20 0.63
NPC1 O15118 1/20 0.63
RAB9A P51151 1/20 0.63
SMN1; SMN2 Q16637 1/20 0.63
RXFP1 Q9HBX9 1/20 0.63
HTT P42858 2/20 0.62
ESR1 P03372 2/20 0.61
POLB P06746 1/20 0.61
DNMT1 P26358 1/20 0.61
LMNA P02545 2/20 0.60
MAPK1 P28482 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22071795 0.85 ALDH1A1 (0.82) ALDH1A1TSHRMAPTCREBBPHSD17B10
SCHEMBL22042856 0.83 TSHR (0.74) ALDH1A1TSHRMAPTCREBBPHSD17B10
SCHEMBL19342077 0.83 ALDH1A1 (0.79) ALDH1A1TSHRMAPTCREBBPHSD17B10
SCHEMBL19342110 0.82 DAPK3 (0.78) ALDH1A1TSHRMAPTCREBBPHSD17B10
SCHEMBL19342064 0.81 TSHR (0.71) ALDH1A1TSHRMAPTCREBBPHSD17B10
SCHEMBL19342093 0.81 L3MBTL1 (0.75) ALDH1A1TSHRMAPTCREBBPHSD17B10
SCHEMBL19342086 0.79 KMT2A (0.81) ALDH1A1TSHRMAPTCREBBPHSD17B10
SCHEMBL22071798 0.78 L3MBTL1 (1.00) ALDH1A1TSHRMAPTCREBBPHSD17B10
SCHEMBL19342080 0.78 ALDH1A1 (0.70) ALDH1A1TSHRMAPTCREBBPHSD17B10
SCHEMBL28782970 0.77 ALDH1A1 (1.00) ALDH1A1TSHRMAPTCREBBPHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3892622-A1 COMPOUNDS HAVING PDE9A INHIBITORY ACTIVITY, AND PHARMACEUTICAL USES THEREOF Korea Research Institute of Chemical Technology (KR) 2021-10-13 EP disclosed