SCHEMBL23924017

SCHEMBL23924017

COc1cc2ncccc2cc1C(N)=O

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 1/20 0.64
PDGFRA P16234 1/20 0.64
KDR P35968 6/20 0.55
AURKA O14965 5/20 0.55
MET P08581 5/20 0.55
TEK Q02763 5/20 0.55
AURKB Q96GD4 5/20 0.55
KDM4E B2RXH2 4/20 0.51
ALDH1A1 P00352 3/20 0.51
HPGD P15428 3/20 0.51
GLA P06280 1/20 0.51
GAA P10253 1/20 0.51
ABL1 P00519 1/20 0.50
LCK P06239 1/20 0.50
LYN P07948 1/20 0.50
MKNK1 Q9BUB5 1/20 0.49
MKNK2 Q9HBH9 1/20 0.49
ALOX15 P16050 1/20 0.48
HTT P42858 1/20 0.48
IRAK4 Q9NWZ3 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29535684 1.00 PDGFRB (0.64) PDGFRBPDGFRAKDRAURKAMET
Hydrochloric Acid SCHEMBL27894607 0.99 PDGFRB (0.62) PDGFRBPDGFRAKDRAURKAMET
SCHEMBL30152477 0.94 PDGFRB (0.64) PDGFRBPDGFRAKDRAURKAMET
SCHEMBL28839474 0.94 PDGFRB (0.64) PDGFRBPDGFRAKDRAURKAMET
SCHEMBL30229311 0.94 PDGFRB (0.64) PDGFRBPDGFRAKDRAURKAMET
SCHEMBL29372253 0.93 PDGFRB (0.56) PDGFRBPDGFRAKDRAURKAMET
SCHEMBL23640270 0.87 PDGFRB (0.66) PDGFRBPDGFRAKDRAURKAKDM4E
SCHEMBL29488239 0.87 PDGFRB (0.66) PDGFRBPDGFRAAURKAKDM4EALDH1A1
SCHEMBL30448935 0.85 PDGFRB (0.64) PDGFRBPDGFRAAURKAKDM4EALDH1A1
SCHEMBL30152708 0.85 PDGFRB (0.49) PDGFRBPDGFRAKDRAURKAMET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115298198-A Novel compounds and compositions for targeted therapy of kidney-related cancers 上海盟科药业股份有限公司 2022-11-04 CN claimed
CN-107266363-A Methanesulfonic acid pleasure is cut down for the preparation method of Buddhist nun's impurity of the drug 杭州华东医药集团新药研究院有限公司 2017-10-20 CN claimed
US-20260083724-A1 COMPOUNDS TARGETING PAX3::FOXO1 FUSION PROTEIN GEORGETOWN UNIVERSITY (US) 2026-03-26 US disclosed
US-12391666-B2 Indoline-1-formamide compound, preparation method therefor, and medical use thereof BEIJING INNOCARE PHARMA TECH CO., LTD. (CN) 2025-08-19 US disclosed
CN-116751162-B Quinoline compound, preparation method thereof, pharmaceutical composition and medical application 中国人民解放军军事科学院军事医学研究院 2025-02-28 CN disclosed
CN-117865887-A Preparation method of lenvatinib mesylate intermediate 山东鲁抗医药股份有限公司 2024-04-12 CN disclosed
CN-117624044-A Preparation method of lenvatinib 山东新时代药业有限公司 2024-03-01 CN disclosed
US-20240043414-A1 Compounds for the Treatment of Kinase-Dependent Disorders EXELIXIS, INC. 2024-02-08 US disclosed
CN-117321036-A phenyl-O-quinoline, quinazoline, thienopyridine, thienopyrimidine, pyrrolopyridine, pyrrolopyrimidine compounds having anticancer activity 成都安泰康赛生物科技有限公司 2023-12-29 CN disclosed
CN-116751161-A Quinoline compound, preparation method thereof, pharmaceutical composition and medical application 中国人民解放军军事科学院军事医学研究院 2023-09-15 CN disclosed
CN-116751162-A Quinoline compound, preparation method thereof, pharmaceutical composition and medical application 中国人民解放军军事科学院军事医学研究院 2023-09-15 CN disclosed
CN-113924288-A Quinolyl-containing compound, pharmaceutical composition and application thereof 北京普祺医药科技有限公司 2022-01-11 CN disclosed
US-20210322404-A1 FGFR REGULATION FOR THE TREATMENT OF VIRAL INFECTIONS ETH ZURICH (CH) 2021-10-21 US disclosed
CN-110003219-A Pyrazolo [1,5A] pyrimidine and thieno [3,2B] pyrimidine derivatives as IRAK4 regulator 弗·哈夫曼-拉罗切有限公司 2019-07-12 CN disclosed
CN-109851556-A Logical sequence cuts down the preparation method for Buddhist nun or its mesylate drug impurity 扬子江药业集团有限公司 2019-06-07 CN disclosed
CN-105367577-B Pyrazolo [1,5A] pyrimidine and thieno [3,2B] pyrimidine derivatives as IRAK4 regulator 弗·哈夫曼-拉罗切有限公司 2019-04-23 CN disclosed
CN-107305202-A The HPLC methods and impurity that analysis methanesulfonic acid pleasure is cut down for Buddhist nun and its preparation impurity make the purposes of reference standard 北京睿创康泰医药研究院有限公司 2017-10-31 CN disclosed
CN-107266363-A Methanesulfonic acid pleasure is cut down for the preparation method of Buddhist nun's impurity of the drug 杭州华东医药集团新药研究院有限公司 2017-10-20 CN disclosed
CN-104876864-B A kind of pleasure cuts down the preparation method for Buddhist nun 北京康立生医药技术开发有限公司 2017-03-08 CN disclosed
CN-105801481-A Lenvatinib synthesizing method 湖南欧亚生物有限公司 2016-07-27 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12391666-B2 Indoline-1-formamide compound, preparation method therefor, and medical use thereof FLT1, KDR, TEK PDGFRB 38/4885PDGFRA 25/4885KDR 2/4885
US-20260083724-A1 COMPOUNDS TARGETING PAX3::FOXO1 FUSION PROTEIN PAX3, FOXO1, PAXBP1 PDGFRB 2327/4885PDGFRA 2497/4885KDR 1973/4885
US-20240043414-A1 Compounds for the Treatment of Kinase-Dependent Disorders ERBB2, MAP3K6, MAP3K1 PDGFRB 327/4885PDGFRA 564/4885KDR 237/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.