Camptothecin

Camptothecin

SCHEMBL23929267

CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3ccccc3nc2-1.O=C(O)CCl

nearest known ligand 0.88

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 18/20 0.88
ALDH1A1 P00352 4/20 0.88
KDM4E B2RXH2 4/20 0.88
MEN1 O00255 4/20 0.88
KMT2A Q03164 4/20 0.88
SMN1; SMN2 Q16637 4/20 0.88
GLA P06280 3/20 0.88
TP53 P04637 2/20 0.88
HPGD P15428 2/20 0.88
CYP3A4 P08684 2/20 0.88
HBB P68871 2/20 0.88
RAB9A P51151 2/20 0.88
BLM P54132 2/20 0.88
STAT6 P42226 1/20 0.88
CHEK1 O14757 1/20 0.88
HDAC3 O15379 1/20 0.88
ABCC4 O15439 1/20 0.88
GMNN O75496 1/20 0.88
LMNA P02545 1/20 0.88
CYP1A2 P05177 1/20 0.88

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Camptothecin SCHEMBL2864815 0.96 TOP1 (0.93) TOP1ALDH1A1KDM4EMEN1KMT2A
Camptothecin SCHEMBL1618774 0.95 TOP1 (0.91) TOP1ALDH1A1KDM4EMEN1KMT2A
Camptothecin SCHEMBL5967412 0.95 TOP1 (0.95) TOP1ALDH1A1KDM4EMEN1KMT2A
Camptothecin SCHEMBL5491504 0.94 TOP1 (0.90) TOP1ALDH1A1KDM4EMEN1KMT2A
Camptothecin SCHEMBL6038 0.94 TOP1 (1.00) TOP1ALDH1A1KDM4EMEN1KMT2A
Camptothecin SCHEMBL2298909 0.94 TOP1 (1.00) TOP1ALDH1A1KDM4EMEN1KMT2A
Camptothecin SCHEMBL29369924 0.94 TOP1 (1.00) TOP1ALDH1A1KDM4EMEN1KMT2A
Camptothecin SCHEMBL788063 0.94 TOP1 (1.00) TOP1ALDH1A1KDM4EMEN1KMT2A
Camptothecin SCHEMBL4304557 0.94 TOP1 (1.00) TOP1ALDH1A1KDM4EMEN1KMT2A
Camptothecin SCHEMBL29351099 0.94 TOP1 (1.00) TOP1ALDH1A1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4168009-A1 CONJUGATES OF A CELL-BINDING MOLECULE WITH CAMPTOTHECIN ANALOGS Hangzhou DAC Biotech Co., Ltd. (CN) 2023-04-26 EP disclosed
CN-115443134-A Conjugates of cell binding molecules and camptothecin analogs 杭州多禧生物科技有限公司 2022-12-06 CN disclosed
WO-2021212638-A1 CONJUGATES OF A CELL-BINDING MOLECULE WITH CAMPTOTHECIN ANALOGS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2021-10-28 WO disclosed