SCHEMBL23935154

SCHEMBL23935154

CS1(N=O)C=C1Cc1nc2c(N)nc3ccc(Cl)cc3c2[nH]1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HTR3A P46098 2/20 0.33
HRH4 Q9H3N8 2/20 0.33
KDM4E B2RXH2 1/20 0.33
TUBB4A P04350 2/20 0.33
TUBB P07437 2/20 0.33
TUBA3C P0DPH7 2/20 0.33
TUBA1B P68363 2/20 0.33
TUBA4A P68366 2/20 0.33
TUBB4B P68371 2/20 0.33
TUBB3 Q13509 2/20 0.33
TUBB2A Q13885 2/20 0.33
TUBB8 Q3ZCM7 2/20 0.33
TUBA3E Q6PEY2 2/20 0.33
TUBA1A Q71U36 2/20 0.33
TUBA1C Q9BQE3 2/20 0.33
TUBB6 Q9BUF5 2/20 0.33
TUBB2B Q9BVA1 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23935193 0.81 GABRA1 (0.35) HTR3AHRH4TUBB4ATUBBTUBA3C
SCHEMBL22814407 0.71 NLRP3 (0.40) ADORA3ADORA2AALDH1A1HTR3AHRH4
SCHEMBL20761866 0.70 NLRP3 (0.60) ADORA3ADORA2AKDM4EPIM1PIM2
SCHEMBL23935156 0.69 GABRA1 (0.35) ALDH1A1TYMSPIM1PIM3
SCHEMBL23935066 0.67 GABRA1 (0.39) ALDH1A1KDM4ETYMSF10
SCHEMBL20761532 0.67 NLRP3 (0.61) ADORA3ADORA2AALDH1A1KDM4EPIM1
SCHEMBL23934984 0.67 LRRK2 (0.35) PIM1
SCHEMBL21949527 0.63 NLRP3 (0.55) ALDH1A1KDM4EPIM1PIM2
SCHEMBL20943755 0.62 TLR7 (0.43) PIM1PIM2
SCHEMBL20761303 0.62 NLRP3 (0.62) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3350178-B1 NOVEL IMIDAZO [4,5-C]QUINOLINE AND IMIDAZO [4,5-C][1,5]NAPHTHYRIDINE DERIVATIVES AS LRRK2 INHIBITORS PFIZER (US) 2021-10-20 EP disclosed