SCHEMBL2393560

SCHEMBL2393560

CC1=Cc2ccccc2N(C)C1(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
GAA P10253 3/20 0.39
LMNA P02545 3/20 0.39
MCL1 Q07820 2/20 0.39
PAX8 Q06710 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KDM4E B2RXH2 6/20 0.34
MAPT P10636 5/20 0.34
HPGD P15428 2/20 0.34
NSD2 O96028 1/20 0.34
APP P05067 1/20 0.34
SNCA P37840 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ATM Q13315 1/20 0.34
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 2/20 0.33
POLB P06746 1/20 0.33
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31395894 1.00 ALDH1A1 (0.39) ALDH1A1GAALMNAMCL1PAX8
SCHEMBL30558752 0.76 GPR84 (0.31) GPR84
SCHEMBL30487691 0.76 GAA (0.36) ALDH1A1GAALMNAMCL1PAX8
SCHEMBL4895528 0.75 ALDH1A1 (0.34) ALDH1A1GAALMNAMCL1PAX8
SCHEMBL29008613 0.71 P2RX4 (0.33)
SCHEMBL5501970 0.71 ALDH1A1 (0.34) ALDH1A1GAALMNAMCL1PAX8
SCHEMBL17275723 0.65 ALDH1A1 (0.50) ALDH1A1GAALMNAMCL1PAX8
SCHEMBL297288 0.65 GAA (0.41) ALDH1A1GAALMNAMCL1PAX8
SCHEMBL30437327 0.65 GAA (0.41) ALDH1A1GAALMNAMCL1PAX8
SCHEMBL31414122 0.64 GAA (0.39) ALDH1A1GAALMNAMCL1PAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101768112-B Two-photon induced luminous compound with symmetrical both ends and synthesis method and purposes thereof CHINESE ACAD INST CHEMISTRY 2012-05-30 CN disclosed
US-8017775-B2 1-2-dihydroquinoline derivative having glucocorticoid receptor binding activity SANTEN PHARMACEUTICAL CO., LTD. (JP) 2011-09-13 US disclosed
CN-101768112-A Two-photon induced luminous compound with symmetrical both ends and synthesis method and purposes thereof CHINESE ACAD INST CHEMISTRY 2010-07-07 CN disclosed
US-20090326009-A1 Novel 1-2-Dihydroquinoline Derivative Having Glucocorticoid Receptor Binding Activity Santen Pharmaceutical Co., (JP) 2009-12-31 US disclosed
WO-2009103007-A2 STEROID HORMONE RECEPTOR MODULATOR COMPOUNDS AND METHODS LIGAND PHARMACEUTICALS INCORPORATED (US) 2009-08-20 WO disclosed
US-4374958-A WIRE OR CABLE WITH PROTECTIVE COATING, CROSSLINKING INHIBITION UNION CARBIDE CORPORATION (US) 1983-02-22 US disclosed
US-4046765-A Dihydroquinoline derivatives of antioxidant activity and a process for the preparation thereof MATERIAL KSZ. (HU) 1977-09-06 US disclosed
US-4025631-A Dihydroquinoline derivatives of antioxidant activity MATERIAL KSZ. (HU) 1977-05-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090326009-A1 Novel 1-2-Dihydroquinoline Derivative Having Glucocorticoid Receptor Binding Activity NR3C1, NR3C2, NR5A1 ALDH1A1 3569/4885GAA 4651/4885LMNA 4519/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.