SCHEMBL23937730

SCHEMBL23937730

CCc1cc2cnn(C)c2nc1C

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
GRM1 Q13255 5/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
ALOX15 P16050 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.32
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32
HTR2C P28335 1/20 0.32
KDM5A P29375 1/20 0.31
KDM4C Q9H3R0 1/20 0.31
CYP11B2 P19099 1/20 0.31
NAMPT P43490 1/20 0.31
APP P05067 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23382294 0.77 MEN1 (0.33) MEN1KMT2ASMN1; SMN2ALOX15KDM4E
SCHEMBL21958547 0.77 GRM1 (0.38) GRM1ALDH1A1
SCHEMBL29750581 0.75 ALDH1A1 (0.37) MEN1KMT2AKDM4EALDH1A1
SCHEMBL17680242 0.74 NOS3 (0.39) NOS3NOS1NOS2
SCHEMBL20674173 0.73 HPGD (0.41) MEN1KMT2AKDM4EALDH1A1APP
SCHEMBL24597613 0.73 ALDH1A1 (0.33) MEN1KMT2AKDM4EALDH1A1APP
SCHEMBL24597614 0.73 TSHR (0.35) MEN1KMT2AKDM4EALDH1A1
SCHEMBL23937882 0.73 GRM1 (0.36) GRM1SMN1; SMN2ALOX15
SCHEMBL22778947 0.70 CACNA1H (0.40) MEN1KMT2ASMN1; SMN2ALOX15KDM4E
SCHEMBL3345735 0.69 USP7 (0.40) NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3399968-B1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LTD (KY) 2021-10-20 EP disclosed