SCHEMBL2393775

SCHEMBL2393775

C[C@H]1CN(Cc2ccc(N(C)C(=O)N3CCC(Nc4ccccc4C(N)=O)CC3)cc2)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.39
FAAH O00519 1/20 0.38
MLNR O43193 4/20 0.37
CYP3A4 P08684 3/20 0.37
ALDH1A1 P00352 2/20 0.37
NPC1 O15118 1/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
RAB9A P51151 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PARP1 P09874 5/20 0.36
HDAC1 Q13547 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
USP30 Q70CQ3 1/20 0.36
FPR3 P25089 1/20 0.35
CCR1 P32246 1/20 0.35
GPR65 Q8IYL9 1/20 0.35
GPR35 Q9HC97 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL377935 0.89 FAAH (0.42) FAAHMLNRCYP3A4PARP1FPR3
SCHEMBL2396378 0.88 MLNR (0.45) BRD4FAAHMLNRCYP3A4ALDH1A1
SCHEMBL377747 0.82 MLNR (0.54) MLNRCYP3A4
SCHEMBL377853 0.82 MLNR (0.52) MLNRCYP3A4ALDH1A1NPC1MAPT
SCHEMBL377479 0.81 MLNR (0.49) MLNRCYP3A4
SCHEMBL2397561 0.79 MLNR (0.44) MLNRCYP3A4ALDH1A1NPC1MAPT
SCHEMBL377798 0.78 KDM4E (0.49) FAAHMLNRCYP3A4ALDH1A1FPR3
SCHEMBL377769 0.78 CCR1 (0.44) MLNRCYP3A4MEN1KMT2AFPR3
SCHEMBL2397555 0.77 MLNR (0.52) MLNRUSP30CCR1
SCHEMBL2393780 0.77 FAAH (0.40) FAAHMLNRCYP3A4ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8012981-B2 Benzylpiperazine derivatives as motilin receptor agonists GLAXO GROUP LIMITED (GB) 2011-09-06 US disclosed