SCHEMBL23937829

SCHEMBL23937829

Cn1c(=O)n(C2CC2)c2ccccc21

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.56
CRBN Q96SW2 1/20 0.56
HSD11B1 P28845 1/20 0.51
CYP3A4 P08684 1/20 0.48
PIK3CA P42336 2/20 0.47
PRKDC P78527 2/20 0.47
SLC6A4 P31645 2/20 0.47
DRD2 P14416 1/20 0.47
HPD P32754 1/20 0.46
SLC6A2 P23975 1/20 0.46
CTSS P25774 5/20 0.46
MTOR P42345 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20861040 0.91 PIK3CA (0.53) DDB1CRBNHSD11B1PIK3CAPRKDC
SCHEMBL2986176 0.88 DDB1 (0.54) DDB1CRBNHSD11B1CYP3A4PIK3CA
Hydrochloric Acid SCHEMBL2858713 0.87 DDB1 (0.52) DDB1CRBNHSD11B1CYP3A4PIK3CA
SCHEMBL14186021 0.84 DRD2 (0.57) HSD11B1CYP3A4PIK3CASLC6A4DRD2
SCHEMBL31211853 0.84 DDB1 (0.52) DDB1CRBNHSD11B1CYP3A4PIK3CA
SCHEMBL2636509 0.82 DDB1 (0.51) DDB1CRBNHSD11B1CYP3A4PIK3CA
SCHEMBL2636510 0.82 DDB1 (0.51) DDB1CRBNHSD11B1CYP3A4PIK3CA
SCHEMBL12893497 0.82 HSD11B1 (0.50) DDB1CRBNHSD11B1CYP3A4SLC6A4
SCHEMBL24405567 0.81 DDB1 (0.50) DDB1CRBNHSD11B1CYP3A4CTSS
SCHEMBL11326674 0.81 CTSS (0.48) DDB1CRBNHSD11B1CYP3A4PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3399968-B1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LTD (KY) 2021-10-20 EP disclosed