SCHEMBL23937872

SCHEMBL23937872

Cc1cc2c(cn1)C=CC2=O

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S100A4 P26447 2/20 0.42
CDC25B P30305 3/20 0.36
IDO1 P14902 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
AKT1 P31749 1/20 0.36
SNCA P37840 1/20 0.36
MAP2K1 Q02750 1/20 0.36
PIN1 Q13526 1/20 0.36
EHMT2 Q96KQ7 1/20 0.36
NSD1 Q96L73 1/20 0.36
EHMT1 Q9H9B1 1/20 0.36
UHRF1 Q96T88 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2A6 P11509 1/20 0.33
PIM1 P11309 1/20 0.33
IL5 P05113 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27554383 0.69 S100A4 (0.39) S100A4CDC25BIDO1MAOAMAOB
SCHEMBL13967835 0.65 CA1 (0.45) S100A4CDC25BIDO1MAOAMAOB
SCHEMBL2434782 0.64 CYP1A2 (0.39) MAOBUHRF1CYP1A2CYP2A6IL5
SCHEMBL3197749 0.61 PIM1 (0.48) S100A4CDC25BIDO1MAOAMAOB
SCHEMBL23088443 0.61 PBRM1 (0.46) UHRF1CYP1A2
SCHEMBL11858854 0.61 S100A4 (0.50) S100A4CDC25BIDO1MAOAMAOB
SCHEMBL23235899 0.60 GABRP (0.55) S100A4CDC25BIDO1MAOAMAOB
SCHEMBL24891186 0.60 UHRF1 (0.35) UHRF1CYP1A2CYP2A6
SCHEMBL1889820 0.60 CA1 (0.50)
SCHEMBL2599222 0.60 S100A4 (1.00) S100A4CDC25BIDO1MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3399968-B1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LTD (KY) 2021-10-20 EP disclosed