SCHEMBL23937899

SCHEMBL23937899

N#Cc1cn(O)c2c1CCCC2

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
CYP2C9 P11712 1/20 0.30
KDM5A P29375 1/20 0.30
KDM5B Q9UGL1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23937917 0.98 HSD17B10 (0.35) HSD17B10KDM4EALDH1A1CASP1CASP7
SCHEMBL20631142 0.96 KDM4E (0.33) HSD17B10KDM4EALDH1A1CASP1CASP7
SCHEMBL23937926 0.81
SCHEMBL23937833 0.79 MAPK1 (0.33) KDM4ECASP1CASP7
SCHEMBL23937907 0.72 ALOX5 (0.33) HSD17B10KDM4EALDH1A1
SCHEMBL16132568 0.72 IMPDH2 (0.39) HSD17B10KDM4EALDH1A1CASP1CASP7
SCHEMBL23937908 0.71 ALOX5 (0.35) KDM4E
SCHEMBL23937643 0.68 KDM4E (0.34) KDM4EALDH1A1CYP2C9
SCHEMBL23937911 0.67 POLB (0.30)
SCHEMBL20631141 0.67 FABP4 (0.39) HSD17B10KDM4ECASP1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3399968-B1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LTD (KY) 2021-10-20 EP disclosed