SCHEMBL23948323

SCHEMBL23948323

Cn1cc(-c2cnn(-c3cnn4ccc(=O)[nH]c34)c2)cn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.38
AURKA O14965 1/20 0.36
TTK P33981 1/20 0.36
AURKB Q96GD4 1/20 0.36
INCENP Q9NQS7 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.36
ACVR1 Q04771 1/20 0.36
BRD4 O60885 2/20 0.35
EPHX2 P34913 1/20 0.34
PRMT5 O14744 2/20 0.34
WDR77 Q9BQA1 2/20 0.34
CREBBP Q92793 2/20 0.34
KDM5B Q9UGL1 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
PDE10A Q9Y233 1/20 0.33
MET P08581 1/20 0.33
AXL P30530 2/20 0.32
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26306213 0.88 KDM5B (0.32) CREBBPKDM5B
SCHEMBL23947980 0.86 HCAR1 (0.35) CREBBPKDM5B
SCHEMBL26306206 0.85
SCHEMBL26306189 0.85 PIK3CD (0.31)
SCHEMBL23948322 0.85 MELK (0.40)
SCHEMBL23948320 0.85 EGLN1 (0.32)
SCHEMBL23948326 0.84 CREBBP (0.34) BRD4CREBBP
SCHEMBL26306173 0.83 ADORA3 (0.33) PRMT5WDR77
SCHEMBL23947973 0.82
SCHEMBL23948325 0.82 FLT3 (0.34) ACVR1MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230242536-A1 METHODS FOR PREPARING TYROSINE RECEPTOR KINASE INHIBITORS PYRAMID BIOSCIENCES, INC. 2023-08-03 US disclosed
WO-2021211882-A1 METHODS FOR PREPARING TYROSINE RECEPTOR KINASE INHIBITORS PYRAMID BIOSCIENCES, INC. (US) 2021-10-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230242536-A1 METHODS FOR PREPARING TYROSINE RECEPTOR KINASE INHIBITORS LTK, FRK, LCK MAPK1 456/4885AURKA 243/4885TTK 16/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.