SCHEMBL23949271

SCHEMBL23949271

CC(C)c1cc(Oc2cc(C#N)ccc2Br)n(C)n1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EIF4E P06730 1/20 0.34
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
AR P10275 3/20 0.32
CYP19A1 P11511 1/20 0.31
FFAR1 O14842 1/20 0.30
ICMT O60725 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23949239 0.83 CYP19A1 (0.33) EIF4EMKNK1MKNK2ARCYP19A1
SCHEMBL30353335 0.83 CYP19A1 (0.33) EIF4EMKNK1MKNK2ARCYP19A1
SCHEMBL23949599 0.80 KMT2A (0.41)
SCHEMBL23949263 0.77 EGLN2 (0.34) EIF4EMKNK1MKNK2
SCHEMBL23949274 0.77 EIF4E (0.31) EIF4EMKNK1MKNK2
SCHEMBL25554407 0.75 NSD2 (0.37) EIF4EMKNK1MKNK2CYP19A1ICMT
SCHEMBL30353072 0.75 NSD2 (0.37) EIF4EMKNK1MKNK2CYP19A1ICMT
SCHEMBL23949264 0.75
SCHEMBL23949272 0.73 CYP19A1 (0.34) EIF4EMKNK1MKNK2CYP19A1ICMT
SCHEMBL30353064 0.73 NSD2 (0.38) EIF4EMKNK1MKNK2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230167073-A1 ARYL OR HETEROARYL DERIVATIVE TEIJIN PHARMA LIMITED (JP) 2023-06-01 US disclosed
CN-115996910-A Aryl or heteroaryl derivatives 帝人制药株式会社 2023-04-21 CN disclosed
EP-4137481-A1 ARYL OR HETEROARYL DERIVATIVE Teijin Pharma Limited (JP) 2023-02-22 EP disclosed
WO-2021210650-A1 ARYL OR HETEROARYL DERIVATIVE 帝人ファーマ株式会社 2021-10-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230167073-A1 ARYL OR HETEROARYL DERIVATIVE ARRB1, NR3C2, TRPC6 EIF4E 2352/4885MKNK1 2249/4885MKNK2 2366/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.