SCHEMBL23957604

SCHEMBL23957604

CC(C)Oc1cc(Oc2ccc(N3c4ccccc4NC3O)cn2)ccc1C#N

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGDR Q13258 1/20 0.34
XDH P47989 1/20 0.32
CYP19A1 P11511 1/20 0.32
AR P10275 1/20 0.32
HRH3 Q9Y5N1 2/20 0.31
S1PR1 P21453 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19670125 0.79 PTGDR (0.37) PTGDRXDHARHRH3IRAK4
SCHEMBL23957566 0.78 HRH3 (0.31) CYP19A1HRH3
SCHEMBL18952980 0.75 PTGDR (0.34) PTGDRXDHARHRH3IRAK4
SCHEMBL1980154 0.73 IRAK4 (0.36) PTGDRXDHARIRAK4
SCHEMBL23926955 0.73 NTRK1 (0.38) PTGDRXDH
SCHEMBL18952992 0.73 MMP13 (0.39) PTGDRXDHAR
SCHEMBL17354624 0.73 AR (0.49) XDHCYP19A1AR
SCHEMBL1980041 0.72 KDM4E (0.48) XDHCYP19A1AR
SCHEMBL1979015 0.71 AR (0.45) PTGDRXDHAR
SCHEMBL13832579 0.70 AR (0.36) PTGDRXDHARIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214090-A1 KV3 ENHANCERS FOR THE TREATMENT OF COGNITIVE DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2021-10-28 WO disclosed