SCHEMBL23958274

SCHEMBL23958274

N=Cc1cccc(Nc2nc3ccccc3c(=O)n2-c2ccccc2)c1O

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.43
MAPT P10636 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
LMNA P02545 2/20 0.43
MEN1 O00255 3/20 0.42
POLB P06746 3/20 0.42
KMT2A Q03164 3/20 0.42
GAA P10253 1/20 0.42
KLK7 P49862 1/20 0.42
PDE7A Q13946 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24089980 0.77 ALDH1A1 (0.51) MAPTSMN1; SMN2MEN1POLBKMT2A
SCHEMBL24110933 0.73 MAPT (0.41) TP53MAPTLMNAPOLBPDE7A
SCHEMBL23958140 0.72 RAB9A (0.43) MAPTLMNAPOLBPDE7A
SCHEMBL24110980 0.72 MAPT (0.45) MAPTPDE7A
SCHEMBL23958271 0.71 MAPT (0.43) MAPTLMNAMEN1POLBKMT2A
SCHEMBL24111019 0.71 MAPT (0.47) TP53MAPTLMNAPOLBPDE7A
SCHEMBL24090010 0.70 USP2 (0.52) MAPTMEN1POLBKMT2APDE7A
SCHEMBL23065087 0.70 PIK3CD (0.47) KMT2APDE7A
SCHEMBL24090012 0.70 TOP2A (0.60) MAPTPOLBPDE7A
SCHEMBL1960453 0.69 TP53 (0.70) TP53MAPTSMN1; SMN2LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021215537-A1 2-HETEROARYLAMINOQUINAZOLINONE DERIVATIVE 大日本住友製薬株式会社 (JP) 2021-10-28 WO disclosed