SCHEMBL23958613

SCHEMBL23958613

COc1cc(C(=O)O)cc(/C=C(\N)C2CC2)c1N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA4 P22748 2/20 0.43
CA6 P23280 2/20 0.43
CA7 P43166 2/20 0.43
CA9 Q16790 2/20 0.43
CA14 Q9ULX7 2/20 0.43
CA3 P07451 1/20 0.43
PKM P14618 1/20 0.43
CA5A P35218 1/20 0.43
CA5B Q9Y2D0 1/20 0.43
TPMT P51580 2/20 0.42
PTGS2 P35354 1/20 0.41
KMT2A Q03164 1/20 0.40
CNR2 P34972 1/20 0.38
HTT P42858 1/20 0.37
KDM4E B2RXH2 1/20 0.36
PDE4A P27815 3/20 0.36
PDE4B Q07343 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958934 0.77 CA12 (0.44) CA12CA1CA2CA4CA6
SCHEMBL10337638 0.74 CA12 (0.67) CA12CA1CA2CA4CA6
SCHEMBL23958597 0.74 KMT2A (0.40) CA12CA1CA2CA4CA6
SCHEMBL21723570 0.70 CA12 (0.60) CA12CA1CA2CA4CA6
SCHEMBL23958596 0.70 MAPT (0.44) CA12CA1CA2CA7CA9
SCHEMBL23958843 0.69 ALDH1A1 (0.33) KMT2AHTTALDH1A1HPGD
SCHEMBL5069164 0.69 CA12 (0.58) CA12CA1CA2CA4CA6
SCHEMBL22458580 0.69 CA12 (0.58) CA12CA1CA2CA4CA6
SCHEMBL18009390 0.67 CA12 (0.56) CA12CA1CA2CA4CA6
SCHEMBL1675754 0.67 HTT (0.59) CA12CA1CA2CA4CA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed