SCHEMBL23958679

SCHEMBL23958679

N#Cc1ccnc(-c2ccc(F)cc2)c1-n1ccc(N)nc1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.37
MAPK13 O15264 2/20 0.37
MAPK12 P53778 2/20 0.37
MAPK11 Q15759 2/20 0.37
CHUK O15111 1/20 0.37
ADORA2A P29274 3/20 0.37
ADORA1 P30542 3/20 0.37
ADORA2B P29275 1/20 0.37
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4D Q08499 1/20 0.36
KCNH2 Q12809 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
CSNK2A1 P68400 1/20 0.34
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
HSD17B10 Q99714 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12490922 0.68 HCAR1 (0.37) MAPK14MAPK13MAPK12MAPK11KCNH2
SCHEMBL23930180 0.66 ERBB2 (0.42) CHUKADORA2AADORA1PDE3BPDE3A
SCHEMBL28988564 0.65 MAOB (0.43) CHUKADORA2AADORA1PDE3BPDE3A
SCHEMBL21283226 0.63 CNR2 (0.50) MAPK14CHUKADORA2AADORA1ADORA2B
SCHEMBL16321240 0.62 ADORA1 (0.71) CHUKADORA2AADORA1ADORA2BCSNK2A1
SCHEMBL22180269 0.60 CHUK (0.46) CHUKADORA2AADORA1ADORA2BCSNK2A1
SCHEMBL21911775 0.60 KDM4C (0.30) KDM4C
SCHEMBL30364487 0.59 FAAH (0.44) MAPK14ADORA2AADORA1ALDH1A1MAPT
SCHEMBL20001703 0.59 ADORA2A (0.33) ADORA2AADORA1ADORA2BALDH1A1KDM4E
SCHEMBL22082173 0.58 PTK2 (0.43) MAPK14ALDH1A1KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed