SCHEMBL23958692

SCHEMBL23958692

COc1cc(C(=O)NCC(c2cc(C(C)C)c(F)c(-c3ccc(F)c(F)c3)n2)C2CC2)cc2cc(C)c(F)nc12

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSA P10619 11/20 0.36
ROCK2 O75116 4/20 0.33
ROCK1 Q13464 4/20 0.33
HPGD P15428 1/20 0.32
GRM5 P41594 1/20 0.31
GRM1 Q13255 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958859 0.81 CFTR (0.34) CTSAROCK2ROCK1ALDH1A1POLB
SCHEMBL23958874 0.78 CTSA (0.35) CTSAROCK2ROCK1HPGD
SCHEMBL23958990 0.78 CFTR (0.33) ROCK2ROCK1ALDH1A1POLB
SCHEMBL25698133 0.78 PDE4B (0.35) ROCK2ROCK1
SCHEMBL30006992 0.72 CTSA (0.35) CTSAROCK2ROCK1
SCHEMBL23958639 0.72 CTSA (0.35) CTSAROCK2ROCK1
SCHEMBL23958805 0.72 CTSA (0.35) CTSAROCK2ROCK1
SCHEMBL25697249 0.72 CETP (0.34) CTSAROCK2ROCK1
SCHEMBL23958966 0.71 GABRA5 (0.33) CTSA
SCHEMBL25698156 0.71 PDE4B (0.34) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed