SCHEMBL23958990

SCHEMBL23958990

COc1cc(C(=O)NCC(c2cc(C(C)(C)O)c(Cl)c(-c3ccc(F)cc3)n2)C2CC2)cc2cc(C)c(F)nc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 3/20 0.33
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
CNR2 P34972 4/20 0.32
CNR1 P21554 2/20 0.32
ALDH1A1 P00352 3/20 0.31
KDM4E B2RXH2 2/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
KCNH2 Q12809 1/20 0.31
MAPT P10636 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ACSS2 Q9NR19 1/20 0.31
DDR1 Q08345 1/20 0.31
ROCK2 O75116 1/20 0.30
ROCK1 Q13464 1/20 0.30
POLB P06746 1/20 0.30
RECQL P46063 1/20 0.30
P2RX7 Q99572 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958859 0.94 CFTR (0.34) CFTRLMNATP53CNR2CNR1
SCHEMBL23958810 0.87 CFTR (0.34) CFTRLMNATP53MAPTSMN1; SMN2
SCHEMBL23958786 0.83 IRAK4 (0.32) CFTRLMNAKCNH2MAPTP2RX7
SCHEMBL25687252 0.82 CFTR (0.34) CFTRCNR2CNR1ALDH1A1KDM4E
SCHEMBL23958782 0.82 CFTR (0.35) CFTRLMNATP53ALDH1A1KDM4E
SCHEMBL23958894 0.81 CFTR (0.34) CFTRLMNATP53ALDH1A1KDM4E
SCHEMBL25697344 0.81 ACSS2 (0.30) ACSS2
SCHEMBL23958776 0.81 LMNA (0.36) CFTRLMNATP53ALDH1A1KCNH2
SCHEMBL23958652 0.81 LMNA (0.33) CFTRLMNATP53CNR2CNR1
SCHEMBL23958797 0.81 CFTR (0.36) CFTRLMNATP53ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed