SCHEMBL23958724

SCHEMBL23958724

CC(C)(O)c1cc(C(=O)CN(Cc2ccccc2)Cc2ccccc2)nc(-c2ccc(I)cc2)c1F

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.35
MMP13 P45452 4/20 0.35
MMP1 P03956 3/20 0.35
MMP2 P08253 2/20 0.33
MMP9 P14780 2/20 0.33
THRB P10828 1/20 0.33
PPARG P37231 3/20 0.32
HDAC4 P56524 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
PPARA Q07869 2/20 0.32
PDK1 Q15118 1/20 0.32
MEP1B Q16820 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
KDM4E B2RXH2 1/20 0.31
CASR P41180 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958823 0.92 MMP13 (0.42) CNR1MMP13MMP1MMP2MMP9
SCHEMBL23958718 0.91 CNR1 (0.44) CNR1MMP13MMP1PPARGPPARA
SCHEMBL30007475 0.73 CFTR (0.41) CNR1KDM4EMAPT
SCHEMBL23958619 0.73 CFTR (0.41) CNR1KDM4EMAPT
SCHEMBL28909146 0.71 MAPT (0.40) MMP13MMP1MMP2MMP9THRB
SCHEMBL30211226 0.69 MAPT (0.37) MMP13MMP1MMP2MMP9THRB
SCHEMBL23958824 0.69 MAPT (0.37) MMP13MMP1MMP2MMP9THRB
SCHEMBL23958842 0.67 MAPT (0.38) MMP13MMP1MMP2MMP9THRB
SCHEMBL23958867 0.63 CFTR (0.32)
SCHEMBL23958693 0.61 CFTR (0.40) CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed