SCHEMBL23958730

SCHEMBL23958730

CC(C)(O)c1c(F)c(-c2ccc(F)cc2)nc(C(CN)C(F)(F)F)c1F

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CFTR P13569 3/20 0.34
BRAF P15056 1/20 0.32
CDK8 P49336 1/20 0.32
CDK5 Q00535 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
MAPK14 Q16539 1/20 0.31
KDM5B Q9UGL1 1/20 0.31
TGFBR1 P36897 2/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
GCGR P47871 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958765 1.00 CFTR (0.34) CFTRBRAFCDK8CDK5CLK4
SCHEMBL23958860 0.80 RPS6KB1 (0.33) CFTRBRAFCDK8CDK5CLK4
SCHEMBL23958800 0.79 KDM5B (0.32) CFTRCDK8CDK5CLK4KDM5B
SCHEMBL23958763 0.77 CFTR (0.40) CFTRKDM4EALDH1A1LMNA
SCHEMBL23958626 0.77 CFTR (0.40) CFTRKDM4EALDH1A1LMNA
SCHEMBL25686730 0.76 CFTR (0.35) CFTRBRAFCDK8CDK5CLK4
SCHEMBL23958689 0.74 CFTR (0.35) CFTRMEN1KMT2ATGFBR1KDM4E
SCHEMBL23958729 0.74 CFTR (0.35) CFTRMEN1KMT2ATGFBR1KDM4E
SCHEMBL23958643 0.74 CFTR (0.35) CFTRMEN1KMT2ATGFBR1KDM4E
SCHEMBL30006775 0.74 CFTR (0.35) CFTRMEN1KMT2ATGFBR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed