SCHEMBL23958800

SCHEMBL23958800

CC(C)(O)c1c(F)c(C(CN)C(F)(F)F)nc(-c2ccc(F)cc2)c1-n1ccc(N)nc1=O

nearest known ligand 0.32

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM5B Q9UGL1 1/20 0.32
CFTR P13569 3/20 0.31
CDK8 P49336 1/20 0.30
CDK5 Q00535 1/20 0.30
CLK4 Q9HAZ1 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958765 0.79 CFTR (0.34) KDM5BCFTRCDK8CDK5CLK4
SCHEMBL23958730 0.79 CFTR (0.34) KDM5BCFTRCDK8CDK5CLK4
SCHEMBL23958763 0.64 CFTR (0.40) CFTRADORA2AADORA1
SCHEMBL23958626 0.64 CFTR (0.40) CFTRADORA2AADORA1
SCHEMBL23958860 0.62 RPS6KB1 (0.33) CFTRCDK8CDK5CLK4
SCHEMBL12490922 0.61 HCAR1 (0.37)
SCHEMBL23958593 0.60 CFTR (0.39) CFTRADORA2AADORA1
SCHEMBL23958679 0.60 MAPK14 (0.37) ADORA2AADORA1
SCHEMBL23958714 0.60 CFTR (0.40) CFTRADORA2AADORA1
SCHEMBL25686730 0.58 CFTR (0.35) KDM5BCFTRCDK8CDK5CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed