SCHEMBL23959097

SCHEMBL23959097

C=C=CCC1(c2ccccc2C)C(=O)Nc2cc(Br)ccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 2/20 0.36
TP53 P04637 2/20 0.35
MAPT P10636 5/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 3/20 0.34
MEN1 O00255 2/20 0.34
PIM3 Q86V86 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
ACHE P22303 1/20 0.32
GAA P10253 4/20 0.32
MGAM O43451 2/20 0.32
SI P14410 2/20 0.32
MGAM2 Q2M2H8 2/20 0.32
ALDH1A1 P00352 3/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
SLC27A2 O14975 1/20 0.32
ADAMTS5 Q9UNA0 1/20 0.32
KDM4E B2RXH2 1/20 0.31
BRD4 O60885 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23959402 1.00 PIM1 (0.36) PIM1TP53MAPTPOLBKMT2A
SCHEMBL23959106 0.87 PIM1 (0.38) PIM1TP53MAPTPOLBKMT2A
SCHEMBL23959009 0.80 PIM1 (0.39) PIM1TP53MAPTPOLBKMT2A
SCHEMBL23959001 0.73 MDM2 (0.43) TP53ACHE
SCHEMBL23959029 0.71 LMNA (0.47) MAPTPOLBKMT2AMEN1GAA
SCHEMBL23959081 0.70 CASP1 (0.39) TP53MAPTKMT2AALDH1A1SMN1; SMN2
SCHEMBL23959108 0.70 CASP1 (0.39) TP53MAPTKMT2AALDH1A1SMN1; SMN2
SCHEMBL1613300 0.65 MEN1 (0.40) PIM1TP53MAPTKMT2AMEN1
SCHEMBL2499492 0.64 BRD4 (0.57) PIM1TP53MAPTPOLBKMT2A
SCHEMBL11829 0.63 MEN1 (0.52) PIM1TP53POLBKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021212974-A1 RACEMIC AND CHIRAL 3-(2,3-BUTADIENYL)OXYINDOLINONE COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 复旦大学 (CN) 2021-10-28 WO disclosed