SCHEMBL23965976

SCHEMBL23965976

CNc1nc2c(OC)c(OCCC(=O)N3CCN(C)CC3)ccc2c(=O)n1C(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
HPGD P15428 2/20 0.39
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
RAB9A P51151 1/20 0.38
PIK3CD O00329 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23965975 0.86 PIK3CB (0.40) CYP1A2CYP3A4CYP2D6CYP2C19HPGD
SCHEMBL23966069 0.81 ALDH1A1 (0.46) HPGDALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL23966144 0.78 PLAU (0.36) CYP1A2CYP3A4HPGDALDH1A1GAA
SCHEMBL24211056 0.78 PIK3CB (0.41) CYP1A2CYP3A4CYP2D6CYP2C19HPGD
SCHEMBL23966071 0.76 ALDH1A1 (0.40) CYP1A2CYP3A4CYP2D6CYP2C19HPGD
SCHEMBL24211133 0.76 PIK3CB (0.40) CYP1A2CYP3A4CYP2D6CYP2C19HPGD
SCHEMBL22183752 0.71 PIK3CB (0.39) KMT2APIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL23966102 0.70 PIK3CB (0.48) HPGDALDH1A1SMN1; SMN2RAB9APIK3CD
SCHEMBL23965930 0.70 HRH3 (0.44) ALDH1A1PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL22183756 0.69 PIK3CB (0.41) KMT2APIK3CDPIK3CAPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3904343-A1 AMINO QUINAZOLINONE, AMINO ISOQUINOLONE DERIVATIVES AND APPLICATION THEREOF Zhejiang University (CN) 2021-11-03 EP disclosed