SCHEMBL23968104

SCHEMBL23968104

N#Cc1ccc(-n2cc(-c3ccc(N4CCSCC4)cc3)cn2)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 2/20 0.42
CDK1 P06493 2/20 0.42
CDK4 P11802 2/20 0.42
CCNB1 P14635 2/20 0.42
CCND1 P24385 2/20 0.42
CCNE1 P24864 2/20 0.42
CDK2 P24941 2/20 0.42
CCND3 P30281 2/20 0.42
CDK7 P50613 2/20 0.42
CDK9 P50750 2/20 0.42
CCNH P51946 2/20 0.42
MNAT1 P51948 2/20 0.42
CDK6 Q00534 2/20 0.42
MELK Q14680 1/20 0.37
MAPKAPK2 P49137 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CHEK1 O14757 1/20 0.35
GRM5 P41594 2/20 0.35
CYP11B1 P15538 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23968097 0.87 MELK (0.39) CCNT1CDK1CDK4CCNB1CCND1
SCHEMBL23968098 0.84 MELK (0.48) MELKNPC1RAB9ACHEK1GRM5
SCHEMBL23968144 0.83 MELK (0.37) MELKRET
SCHEMBL23968008 0.81 MELK (0.41) CDK1CDK4CCNB1CCND1CCNE1
SCHEMBL23968021 0.79 MELK (0.37) MELKRETKDM4ETP53
SCHEMBL23968116 0.79 MELK (0.39) MELKRET
SCHEMBL23968184 0.78 MELK (0.39) MELKRETAXL
SCHEMBL23968093 0.75 MAP4K4 (0.54) MELKNPC1RAB9A
SCHEMBL23968162 0.74 MELK (0.40) MELKNPC1RAB9AKDM4ELGMN
SCHEMBL23968094 0.74 MELK (0.40) MELKRET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3104705-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2021-11-03 EP disclosed