SCHEMBL23968144

SCHEMBL23968144

N#Cc1cc(Cl)ccc1-n1cc(-c2ccc(N3CCSCC3)cc2)cn1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MELK Q14680 1/20 0.37
MAP4K4 O95819 1/20 0.37
RET P07949 7/20 0.37
AKR1C3 P42330 1/20 0.34
P2RX3 P56373 1/20 0.33
P2RX2 Q9UBL9 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
HSD17B10 Q99714 1/20 0.33
BMP4 P12644 1/20 0.33
CRHR1 P34998 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23968021 0.87 MELK (0.37) MELKRET
SCHEMBL23968116 0.87 MELK (0.39) MELKRETP2RX3P2RX2GAA
SCHEMBL23968184 0.84 MELK (0.39) MELKRET
SCHEMBL23968104 0.83 CCNT1 (0.42) MELKRET
SCHEMBL23968094 0.81 MELK (0.40) MELKRET
SCHEMBL23968093 0.80 MAP4K4 (0.54) MELKMAP4K4AKR1C3MAPT
SCHEMBL23968097 0.79 MELK (0.39) MELKRETHSD17B10
SCHEMBL23968007 0.78 ALDH1A1 (0.44) MELKMAP4K4AKR1C3MAPT
SCHEMBL23968098 0.77 MELK (0.48) MELKMAP4K4RET
SCHEMBL23968008 0.76 MELK (0.41) MELKMAP4K4MAPTCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3104705-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2021-11-03 EP disclosed