SCHEMBL23968116

SCHEMBL23968116

Cc1ccc(-n2cc(-c3ccc(N4CCSCC4)cc3)cn2)c(C#N)c1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MELK Q14680 1/20 0.39
RET P07949 12/20 0.39
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
HSD17B10 Q99714 1/20 0.35
P2RX3 P56373 1/20 0.35
P2RX2 Q9UBL9 1/20 0.35
LRRK2 Q5S007 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23968144 0.87 MELK (0.37) MELKRETGAAMAPTHSD17B10
SCHEMBL23968021 0.87 MELK (0.37) MELKRET
SCHEMBL23968184 0.84 MELK (0.39) MELKRET
SCHEMBL23968097 0.83 MELK (0.39) MELKRETHSD17B10
SCHEMBL23968104 0.79 CCNT1 (0.42) MELKRET
SCHEMBL23968094 0.78 MELK (0.40) MELKRETLRRK2
SCHEMBL23968098 0.77 MELK (0.48) MELKRET
SCHEMBL23968162 0.74 MELK (0.40) MELKGAAMAPTHSD17B10
SCHEMBL23968008 0.71 MELK (0.41) MELKMAPT
SCHEMBL23968179 0.71 GRM4 (0.44) MELK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3104705-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2021-11-03 EP disclosed