SCHEMBL23968111

SCHEMBL23968111

O=C(c1ccc(-c2cnn(-c3ccc(F)cc3)c2)cc1)N1CCC(O)CC1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 2/20 0.51
HSD11B1 P28845 6/20 0.50
SLC6A7 Q99884 2/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
PTPN1 P18031 1/20 0.49
KDM4E B2RXH2 2/20 0.46
POLB P06746 1/20 0.46
GAA P10253 1/20 0.46
MAP4K4 O95819 1/20 0.46
ALDH1A1 P00352 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
ENPP2 Q13822 1/20 0.44
MAPKAPK2 P49137 1/20 0.44
MGLL Q99685 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8160698 0.84 HSD11B1 (0.66) HTR2BHSD11B1SLC6A7MEN1KMT2A
SCHEMBL23968059 0.82 SLC6A7 (0.50) HSD11B1SLC6A7MEN1KMT2APTPN1
SCHEMBL30967272 0.80 HSD11B1 (0.71) HSD11B1MEN1KMT2APTPN1KDM4E
SCHEMBL23967996 0.78 MEN1 (0.43) HTR2BSLC6A7MEN1KMT2AMAP4K4
SCHEMBL180639 0.78 BCL2L1 (0.59) HSD11B1MEN1KMT2AMAP4K4ALDH1A1
SCHEMBL8155644 0.75 HSD11B1 (0.54) HTR2BHSD11B1SLC6A7MEN1KMT2A
SCHEMBL24018950 0.73 HTR2B (0.51) HTR2BHSD11B1SLC6A7MEN1KMT2A
SCHEMBL3641180 0.72 GRM5 (0.76) HSD11B1MEN1KMT2AKDM4EPOLB
SCHEMBL13952174 0.72 HSD11B1 (0.57) HSD11B1SLC6A7MEN1KMT2APTPN1
SCHEMBL21472163 0.72 GRM5 (0.57) HSD11B1MEN1KMT2AALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3104705-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2021-11-03 EP disclosed