SCHEMBL23967996

SCHEMBL23967996

O=C1CN(C(=O)c2ccc(-c3cnn(-c4ccc(F)cc4)c3)cc2)CCN1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
RAB9A P51151 1/20 0.43
SLC6A7 Q99884 2/20 0.43
MAP4K4 O95819 1/20 0.43
LMNA P02545 1/20 0.42
TACR3 P29371 1/20 0.41
MAPKAPK2 P49137 1/20 0.41
HTR2B P41595 2/20 0.41
HRH3 Q9Y5N1 1/20 0.41
JAK2 O60674 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
USP7 Q93009 1/20 0.40
MKNK1 Q9BUB5 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
KDM1A O60341 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21170645 0.82 HRH3 (0.54) MEN1KMT2ARAB9ALMNATACR3
SCHEMBL23968111 0.78 HTR2B (0.51) MEN1KMT2ASLC6A7MAP4K4MAPKAPK2
SCHEMBL23968059 0.77 SLC6A7 (0.50) MEN1KMT2ASLC6A7MAP4K4LMNA
SCHEMBL24018903 0.75 KMT2A (0.46) MEN1KMT2ARAB9ASLC6A7TACR3
SCHEMBL180639 0.74 BCL2L1 (0.59) MEN1KMT2ARAB9AMAP4K4MAPKAPK2
SCHEMBL25205366 0.70 PTGDR2 (0.44) MEN1KMT2ARAB9A
SCHEMBL12093445 0.69 PKM (0.67) MEN1KMT2ARAB9ALMNATACR3
SCHEMBL4751256 0.69 HSP90AA1 (0.55) KMT2ARAB9AHRH3SMN1; SMN2
SCHEMBL14117676 0.69 HRH3 (0.54) MEN1KMT2ARAB9AHRH3JAK2
SCHEMBL623354 0.69 POLB (0.57) MEN1KMT2ARAB9ALMNAHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3104705-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2021-11-03 EP disclosed