SCHEMBL23969858

SCHEMBL23969858

O=CNc1ccc(-c2cc(-c3ccncc3)cc(-c3ccncc3)c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
ERN1 O75460 2/20 0.43
LMNA P02545 2/20 0.42
MAPT P10636 1/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
PSEN1 P49768 1/20 0.41
PSEN2 P49810 1/20 0.41
APH1B Q8WW43 1/20 0.41
NCSTN Q92542 1/20 0.41
APH1A Q96BI3 1/20 0.41
PSENEN Q9NZ42 1/20 0.41
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
LIMK1 P53667 2/20 0.39
CYP17A1 P05093 1/20 0.39
CYP21A2 P08686 1/20 0.39
CYP11B1 P15538 1/20 0.39
QDPR P09417 1/20 0.38
PDE3B Q13370 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11179661 0.94 ALDH1A1 (0.48) ALDH1A1ERN1LMNAMAPTCYP3A4
Hydrochloric Acid SCHEMBL11198973 0.92 ALDH1A1 (0.46) ALDH1A1ERN1LMNAMAPTCYP3A4
SCHEMBL183576 0.81
SCHEMBL23969869 0.80 ALDH1A1 (0.64) ALDH1A1LMNAMAPTLIMK1CNR1
SCHEMBL11194081 0.78 CNR1 (0.50) ALDH1A1ERN1LMNAMAPTHDAC1
SCHEMBL23969769 0.76 ERN1 (0.50) ALDH1A1ERN1CYP3A4CYP17A1CYP11B1
SCHEMBL19270240 0.76 MAPT (0.73) ERN1LMNAMAPTHDAC1HDAC6
SCHEMBL13907332 0.76 MAPT (0.73) ERN1LMNAMAPTHDAC1HDAC6
SCHEMBL13907285 0.76 MAPT (0.73) ERN1LMNAMAPTHDAC1HDAC6
SCHEMBL18748287 0.76 MAPT (0.73) ERN1LMNAMAPTHDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3353156-B1 TEAD TRANSCRIPTION FACTOR AUTOPALMITOYLATION INHIBITORS MASSACHUSETTS GEN HOSPITAL (US) 2021-11-03 EP disclosed