SCHEMBL23969769

SCHEMBL23969769

O=CNc1ccc(-c2cccc(-c3cccnc3)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.50
MKNK1 Q9BUB5 6/20 0.47
MKNK2 Q9HBH9 6/20 0.47
MEN1 O00255 1/20 0.47
PSIP1 O75475 1/20 0.47
AXL P30530 1/20 0.47
CYP2A6 P11509 2/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
KDR P35968 2/20 0.47
CNR1 P21554 1/20 0.47
KMO O15229 1/20 0.46
CYP11B2 P19099 3/20 0.46
CYP11B1 P15538 2/20 0.46
CYP17A1 P05093 1/20 0.46
CYP19A1 P11511 1/20 0.46
PGR P06401 1/20 0.46
EPHX2 P34913 1/20 0.44
PRMT6 Q96LA8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2654544 0.87 CNR1 (0.52) ERN1MKNK1MKNK2MEN1PSIP1
SCHEMBL14425482 0.77 CYP11B2 (0.66) MKNK1MKNK2MEN1PSIP1AXL
SCHEMBL14425488 0.77 CYP11B2 (0.66) MKNK1MKNK2MEN1PSIP1AXL
SCHEMBL12103445 0.77 CYP2A6 (0.79) MKNK1MKNK2MEN1PSIP1AXL
SCHEMBL30620885 0.77 CYP2A6 (0.79) MKNK1MKNK2MEN1PSIP1AXL
SCHEMBL17951830 0.77 CYP2A6 (0.79) MKNK1MKNK2MEN1PSIP1AXL
SCHEMBL23969858 0.76 ALDH1A1 (0.43) ERN1MEN1ALDH1A1CYP3A4CNR1
SCHEMBL17721072 0.76 CYP11B2 (0.63) MKNK1MKNK2MEN1PSIP1AXL
SCHEMBL23969869 0.76 ALDH1A1 (0.64) ALDH1A1CNR1PGR
SCHEMBL18134278 0.76 CYP11B2 (0.63) MKNK1MKNK2MEN1PSIP1AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3353156-B1 TEAD TRANSCRIPTION FACTOR AUTOPALMITOYLATION INHIBITORS MASSACHUSETTS GEN HOSPITAL (US) 2021-11-03 EP disclosed