SCHEMBL23970889

SCHEMBL23970889

CCCc1nc2ccccc2cc1C(C)C

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 11/20 0.44
ALDH1A1 P00352 3/20 0.42
HPGD P15428 2/20 0.42
GLA P06280 1/20 0.42
MAPT P10636 1/20 0.42
ACHE P22303 1/20 0.42
LCK P06239 1/20 0.41
KDM4E B2RXH2 2/20 0.41
GAA P10253 2/20 0.41
ATM Q13315 1/20 0.39
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
GPBAR1 Q8TDU6 1/20 0.38
CYSLTR1 Q9Y271 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28609423 0.79 TLR8 (0.54) TLR8ALDH1A1HPGDGLAMAPT
SCHEMBL19260213 0.79 TDP1 (0.52) TLR8ALDH1A1HPGDGLAMAPT
Ammonia Solution, Strong SCHEMBL9131397 0.77 TLR8 (0.53) TLR8ALDH1A1HPGDGLAMAPT
SCHEMBL27851831 0.75 KDM4E (0.54) ALDH1A1HPGDMAPTLCKKDM4E
SCHEMBL12388168 0.74 ALDH1A1 (0.55) TLR8ALDH1A1HPGDGLAMAPT
SCHEMBL12410896 0.74 ALDH1A1 (0.48) TLR8ALDH1A1HPGDGLAMAPT
SCHEMBL13949449 0.73 ALOX15 (0.42) TLR8ALDH1A1HPGDGLAMAPT
SCHEMBL2630610 0.73 TLR8 (0.46) TLR8ALDH1A1HPGDGLAMAPT
SCHEMBL14726026 0.73 HPGD (0.48) TLR8ALDH1A1HPGDGLAMAPT
SCHEMBL22045308 0.73 TLR8 (0.57) TLR8ALDH1A1HPGDGLAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222353-A1 MACROCYCLIC INHIBITORS OF PEPTIDYLARGININE DEIMINASES GILEAD SCIENCES, INC. (US) 2021-11-04 WO disclosed