SCHEMBL23970967

SCHEMBL23970967

Nc1nc(Cl)c(F)cc1I

nearest known ligand 0.44

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KHK P50053 1/20 0.44
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30410994 1.00 KHK (0.44) KHKKEAP1NFE2L2
SCHEMBL21223861 0.79 KHK (0.39) KHK
SCHEMBL8237996 0.79 KEAP1 (0.47) KHKKEAP1NFE2L2
SCHEMBL443877 0.79 KHK (0.35) KHK
SCHEMBL34467639 0.79 KEAP1 (0.47) KHKKEAP1NFE2L2
SCHEMBL5925804 0.77 CA1 (0.31) KHK
SCHEMBL24850172 0.77 KHK (0.34) KHK
SCHEMBL31453136 0.74 KEAP1 (0.38) KHKKEAP1NFE2L2
SCHEMBL23030325 0.74 KHK (0.44) KHKKEAP1NFE2L2
SCHEMBL20455590 0.74 ALDH1A1 (0.34) KHK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222353-A1 MACROCYCLIC INHIBITORS OF PEPTIDYLARGININE DEIMINASES GILEAD SCIENCES, INC. (US) 2021-11-04 WO disclosed