SCHEMBL23973019

SCHEMBL23973019

O=C(Cc1ccccc1)N1CCc2nc(C3(c4ccccc4)CC3)[nH]c(=O)c2C1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MTHFD2 P13995 8/20 0.46
KDR P35968 1/20 0.42
OPRD1 P41143 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
CRBN Q96SW2 1/20 0.41
ROCK2 O75116 1/20 0.41
CLPP Q16740 1/20 0.40
KCNK3 O14649 1/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23973188 0.93 CLPP (0.44) MTHFD2KDROPRD1ROCK2CLPP
SCHEMBL23973473 0.92 MTHFD2 (0.42) MTHFD2KDRROCK2CLPP
SCHEMBL23972409 0.92 TRPV1 (0.48) MTHFD2KDRROCK2CLPP
SCHEMBL23972215 0.91 CLPP (0.47) MTHFD2KDROPRD1KMT2AMEN1
SCHEMBL26672609 0.91 MTHFD2 (0.41) MTHFD2KDRROCK2
SCHEMBL23973478 0.91 ROCK2 (0.43) MTHFD2KDROPRD1ROCK2
SCHEMBL23972655 0.91 AURKA (0.42) MTHFD2KDRROCK2CLPP
SCHEMBL23972465 0.91 CLPP (0.46) MTHFD2KDRROCK2CLPP
SCHEMBL26672604 0.91 CLPP (0.45) MTHFD2KDRCLPPKCNK3
SCHEMBL23972407 0.89 MEN1 (0.46) MTHFD2KMT2AMEN1CLPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021221169-A1 PYRIMIDIN-4(3H)-ONE DERIVATIVES AS TRPV4 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2021-11-04 WO disclosed