SCHEMBL2397343

SCHEMBL2397343

NS(=O)(=O)c1ccccc1Cc1c(F)c(F)c(F)c(F)c1F

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA2 P00918 14/20 0.45
CA1 P00915 13/20 0.45
CA9 Q16790 6/20 0.42
CA12 O43570 4/20 0.42
CA7 P43166 4/20 0.42
CA6 P23280 3/20 0.42
CA4 P22748 2/20 0.42
CA5A P35218 2/20 0.42
CA5B Q9Y2D0 2/20 0.42
CYP2C9 P11712 1/20 0.42
CA14 Q9ULX7 1/20 0.42
PTGES2 Q9H7Z7 5/20 0.40
CA13 Q8N1Q1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4664484 0.80 LMNA (0.46) CA2CA1CA9CA12CA7
SCHEMBL4663042 0.77 KCNA5 (0.43) CA2CA1CA9CA12CA7
SCHEMBL7207427 0.76 CA2 (0.41) CA2CA1CA9CA12CA7
SCHEMBL30988956 0.76 CA2 (0.50) CA2CA1CA9CA12CA7
SCHEMBL407413 0.76 CA2 (0.50) CA2CA1CA9CA12CA7
SCHEMBL3651546 0.75 CA2 (0.50) CA2CA1CA9CA12CA7
SCHEMBL31471001 0.75 CA2 (0.50) CA2CA1CA9CA12CA7
SCHEMBL8349565 0.74 CA2 (0.54) CA2CA1CA9CA12CA7
Methane SCHEMBL28850761 0.74 CA2 (0.49) CA2CA1CA9CA12CA7
Hydrochloric Acid SCHEMBL3517386 0.74 CA1 (0.49) CA2CA1CA9CA12CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110212920-A1 N-Substituted Benzene Sulfonamides NEITZEL MARTIN 2011-09-01 US disclosed
US-7208488-B2 N-substituted benzene sulfonamides ELAN PHARMACEUTICALS, INC. (US) 2007-04-24 US disclosed
US-20050165003-A1 Treating Alzheimer's Disease; 4-Chloro-N-(4-hydroxy-3-methoxy-benzyl)-N-(2-oxo-azepan-3-yl)-benzenesulfonamide for example; gamma secretase inhibitors; inhibition of beta-amyloid synthesis with minimal inhibition of Notch Signaling ELAN PHARMACEUTICALS, INC. 2005-07-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050165003-A1 Treating Alzheimer's Disease; 4-Chloro-N-(4-hydroxy-3-methoxy-benzyl)-N-(2-oxo-azepan-3-yl)-benzenesulfonamide for example; gamma secretase inhibitors; inhibition of beta-amyloid synthesis with minimal inhibition of Notch Signaling BACE1, PSEN1, BACE2 CA2 3100/4885CA1 839/4885CA9 2745/4885
US-20110212920-A1 N-Substituted Benzene Sulfonamides PSEN1, PSEN2, BACE1 CA2 3239/4885CA1 591/4885CA9 3047/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.