SCHEMBL23976292

SCHEMBL23976292

COC(=O)C(CCC(C)(C)N)NC(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 10/20 0.43
CTSS P25774 7/20 0.43
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
HTT P42858 1/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
CTSL P07711 2/20 0.40
CTSB P07858 1/20 0.40
KLK5 Q9Y337 1/20 0.39
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
CA12 O43570 1/20 0.38
CA14 Q9ULX7 1/20 0.38
GSTP1 P09211 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5828772 0.92 CTSK (0.48) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL6354784 0.89 CTSK (0.46) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL24299005 0.89 CTSK (0.46) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL24021111 0.87 CTSK (0.39) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL29062803 0.87 CTSK (0.39) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL31341213 0.86 CTSK (0.43) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL24324050 0.84 CTSK (0.43) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL18109360 0.84 CTSK (0.43) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL18109361 0.84 CTSK (0.43) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL2845919 0.84 CTSK (0.44) CTSKCTSSCYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222483-A1 METHODS OF USE FOR PYRIMIDINES AS FERROPORTIN INHIBITORS GLOBAL BLOOD THERAPEUTICS, INC. (US) 2021-11-04 WO disclosed
WO-2021222363-A1 CYCLOALKYL PYRIMIDINES AS FERROPORTIN INHIBITORS GLOBAL BLOOD THERAPEUTICS, INC. (US) 2021-11-04 WO disclosed