SCHEMBL23977102

SCHEMBL23977102

CCc1c(OC)cc(C(=O)OCC(CC)(c2ccccc2)N(C)C)cc1OC

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.81
OPRD1 P41143 2/20 0.81
SLC6A3 Q01959 2/20 0.81
NR1I2 O75469 1/20 0.81
CHRM2 P08172 1/20 0.81
ADORA3 P0DMS8 1/20 0.81
ADRA2B P18089 1/20 0.81
SLC6A4 P31645 1/20 0.81
OPRK1 P41145 1/20 0.81
CHRNA4 P43681 1/20 0.81
PDE4D Q08499 1/20 0.81
KCNH2 Q12809 1/20 0.81
MAPK1 P28482 3/20 0.74
SMN1; SMN2 Q16637 3/20 0.74
MAPT P10636 3/20 0.74
HIF1A Q16665 2/20 0.74
ALDH1A1 P00352 2/20 0.74
MEN1 O00255 2/20 0.74
KMT2A Q03164 2/20 0.74
CYP3A4 P08684 2/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trimebutine SCHEMBL14273976 0.90 OPRM1 (1.00) OPRM1OPRD1SLC6A3NR1I2CHRM2
Trimebutine SCHEMBL25705 0.90 OPRM1 (1.00) OPRM1OPRD1SLC6A3NR1I2CHRM2
Trimebutine SCHEMBL7428847 0.89 OPRM1 (0.98) OPRM1OPRD1SLC6A3NR1I2CHRM2
SCHEMBL16522145 0.86 OPRM1 (0.88) OPRM1OPRD1SLC6A3NR1I2CHRM2
Trimebutine SCHEMBL5011979 0.85 ALDH1A1 (1.00) OPRM1OPRD1SLC6A3NR1I2CHRM2
Trimebutine SCHEMBL67225 0.85 ALDH1A1 (1.00) OPRM1OPRD1SLC6A3NR1I2CHRM2
Trimebutine SCHEMBL1652810 0.85 ALDH1A1 (1.00) OPRM1OPRD1SLC6A3NR1I2CHRM2
Trimebutine SCHEMBL28274910 0.85 ALDH1A1 (1.00) OPRM1OPRD1SLC6A3NR1I2CHRM2
SCHEMBL31432918 0.81 OPRM1 (0.69) OPRM1OPRD1SLC6A3NR1I2CHRM2
SCHEMBL14317655 0.81 OPRM1 (0.83) OPRM1OPRD1SLC6A3NR1I2CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021221544-A1 NOVEL COMPOUND [2-(DIMETHYLAMINO)-2-PHENYLBUTYL]-3,4,5-TRIMETHOXYBENZOATE 4-METHYL-2Н-CHROMEN-2-ON-7-YL SULPHATE AND USE THEREOF ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ВАЛЕНТА-ИНТЕЛЛЕКТ" (RU) 2021-11-04 WO disclosed