SCHEMBL23978902

SCHEMBL23978902

C=C/C=C(\N)c1c(Cl)cc(C(=C)NCc2cccc(F)c2)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.39
NTRK1 P04629 2/20 0.38
PTPN7 P35236 2/20 0.36
DUSP3 P51452 2/20 0.36
DPP4 P27487 1/20 0.36
CNR1 P21554 1/20 0.35
ALOX5 P09917 1/20 0.35
SRC P12931 1/20 0.35
MAPK1 P28482 2/20 0.34
RAB9A P51151 1/20 0.34
GRIN2B Q13224 1/20 0.34
APP P05067 1/20 0.34
P2RY12 Q9H244 1/20 0.34
ROCK2 O75116 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23979015 0.79 EPHX2 (0.44) EPHX2NTRK1PTPN7DUSP3DPP4
SCHEMBL23978774 0.68 MEN1 (0.50) EPHX2SRCROCK2
SCHEMBL23978714 0.67 CYP19A1 (0.35) P2RY12
SCHEMBL23978863 0.67 NPC1 (0.41) RAB9A
SCHEMBL23979115 0.66 TXNRD1 (0.36) P2RY12ROCK2
SCHEMBL23978773 0.65 EPHX2 (0.49) EPHX2P2RY12ROCK2
SCHEMBL23978881 0.65 MEN1 (0.50) PTPN7DUSP3
M-Fluorobenzylguanidine SCHEMBL4335223 0.65 SRC (0.49) PTPN7DUSP3SRCMAPK1RAB9A
SCHEMBL5528698 0.65 PTPN7 (0.50) PTPN7DUSP3SRCMAPK1RAB9A
SCHEMBL31173724 0.65 SRC (0.56) EPHX2SRCMAPK1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed