SCHEMBL23979115

SCHEMBL23979115

C=C(NCc1cccc(CC)c1)c1cc(Cl)c(C(=C)OC)c(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TXNRD1 Q16881 1/20 0.36
TSHR P16473 2/20 0.36
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
HTT P42858 1/20 0.35
MMP13 P45452 1/20 0.35
LMNA P02545 3/20 0.34
HPGD P15428 2/20 0.34
CYP19A1 P11511 1/20 0.34
ROCK2 O75116 1/20 0.33
APEX1 P27695 1/20 0.33
P2RY12 Q9H244 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
ALOX12 P18054 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23978714 0.86 CYP19A1 (0.35) TXNRD1ALDH1A1LMNAHPGDCYP19A1
SCHEMBL23978863 0.76 NPC1 (0.41) APEX1MAPTALOX12
SCHEMBL23979015 0.74 EPHX2 (0.44) P2RY12
SCHEMBL23978881 0.74 MEN1 (0.50) LMNAHPGD
SCHEMBL23979023 0.71 ERCC1 (0.45) ROCK2
SCHEMBL16442463 0.70 LOXL2 (0.49) ALDH1A1SMN1; SMN2HTTLMNAMAPT
SCHEMBL23978902 0.66 EPHX2 (0.39) ROCK2P2RY12
SCHEMBL23978689 0.66 NPC1 (0.55) MMP13HPGDROCK2APEX1
SCHEMBL23978695 0.65 ROCK2 (0.51) SMN1; SMN2HTTMMP13LMNAHPGD
SCHEMBL14581253 0.64 SMN1; SMN2 (0.43) ALDH1A1SMN1; SMN2HTTLMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed